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Evaluating in vivo data for drug metabolism and transport: lessons from Kirchhoff's Laws. Front Pharmacol. 2024; 15:1456677.
Benet LZ, Sodhi JK. PMID: 39564109; PMCID: PMC11574206.
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Is there a possibility that P-glycoprotein reduces reproductive toxicity in males but breast cancer resistance protein does not? Clin Transl Sci. 2024 Oct; 17(10):e70027.
Yu Z, Liu W, Wang Z, Chen Y, Yan J, Benet LZ, Zhai S. PMID: 39356462; PMCID: PMC11446187.
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PubMed Mentions:
1 Fields:
Translation:
HumansAnimals
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Commentary: Pharmacokinetic Theory Must Consider Published Experimental Data. Drug Metab Dispos. 2024 Aug 14; 52(9):932-938.
Benet LZ, Sodhi JK. PMID: 38942444; PMCID: PMC11331591.
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PubMed Mentions:
1 Fields:
Translation:
HumansAnimals
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The potential of developing high hepatic clearance drugs via controlled release: Lessons from Kirchhoff's Laws. J Control Release. 2024 Sep; 373:564-567.
Benet LZ, Tiitto MV, Sodhi JK. PMID: 39032574.
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Translation:
Humans
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Are all measures of liver Kpuu a function of FH, as determined following oral dosing, or have we made a critical error in defining hepatic drug clearance? Eur J Pharm Sci. 2024 May 01; 196:106753.
Benet LZ, Sodhi JK. PMID: 38522769.
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PubMed Mentions:
2 Fields:
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An Explanation of Why Dose-Corrected Area Under the Curve for Alternate Administration Routes Can Be Greater than for Intravenous Dosing. AAPS J. 2024 01 30; 26(1):22.
Wakuda H, Xiang Y, Sodhi JK, Uemura N, Benet LZ. PMID: 38291293.
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PubMed Mentions:
2 Fields:
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Solubility-Permeability Interplay in Facilitating the Prediction of Drug Disposition Routes, Extent of Absorption, Food Effects, Brain Penetration and Drug Induced Liver Injury Potential. J Pharm Sci. 2023 09; 112(9):2326-2331.
Benet LZ. PMID: 37429358; PMCID: PMC11033615.
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PubMed Mentions: Fields:
Translation:
Humans
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The Uses and Advantages of Kirchhoff's Laws vs. Differential Equations in Pharmacology, Pharmacokinetics, and (Even) Chemistry. AAPS J. 2023 04 10; 25(3):38.
Benet LZ, Sodhi JK. PMID: 37038013; PMCID: PMC10832327.
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PubMed Mentions:
4 Fields:
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Using an animal model to predict the effective human dose for oral multiple sclerosis drugs. Clin Transl Sci. 2023 03; 16(3):467-477.
Liu W, Yu Z, Wang Z, Waubant EL, Zhai S, Benet LZ. PMID: 36419359; PMCID: PMC10014696.
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PubMed Mentions:
3 Fields:
Translation:
HumansAnimals
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Review of the application of Kirchhoff's Laws of series and parallel flows to pharmacology: Defining organ clearance. Pharmacol Ther. 2022 Nov; 239:108278.
Pachter JA, Dill KA, Sodhi JK, Benet LZ. PMID: 36075300; PMCID: PMC10832328.
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PubMed Mentions:
4 Fields:
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State of the Art and Uses for the Biopharmaceutics Drug Disposition Classification System (BDDCS): New Additions, Revisions, and Citation References. AAPS J. 2022 02 23; 24(2):37.
Bocci G, Oprea TI, Benet LZ. PMID: 35199251; PMCID: PMC8865883.
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PubMed Mentions:
16 Fields:
Translation:
Animals
-
Does Addition of Protein to Hepatocyte or Microsomal In Vitro Incubations Provide a Useful Improvement in In Vitro-In Vivo Extrapolation Predictability? Drug Metab Dispos. 2022 04; 50(4):401-412.
Kameyama T, Sodhi JK, Benet LZ. PMID: 35086847; PMCID: PMC11022888.
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PubMed Mentions:
1 Fields:
Translation:
Cells
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Can In Vitro-In Vivo Extrapolation Be Successful? Recognizing the Incorrect Clearance Assumptions. Clin Pharmacol Ther. 2022 05; 111(5):1022-1035.
Benet LZ, Sodhi JK. PMID: 34731496; PMCID: PMC9542026.
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PubMed Mentions:
9 Fields:
Translation:
HumansCells
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Analyzing Potential Intestinal Transporter Drug-Drug Interactions: Reevaluating Ticagrelor Interaction Studies. Pharm Res. 2021 Oct; 38(10):1639-1644.
Liu S, Sodhi JK, Benet LZ. PMID: 34729703; PMCID: PMC9595044.
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PubMed Mentions:
4 Fields:
Translation:
HumansAnimals
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Batch Selection via In Vitro/In Vivo Correlation in Pharmacokinetic Bioequivalence Testing. AAPS PharmSciTech. 2021 Aug 19; 22(7):224.
Burmeister Getz E, Carroll KJ, Mielke J, Jones B, Benet LZ. PMID: 34410534.
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PubMed Mentions:
2 Fields:
Translation:
Humans
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Examination of Urinary Excretion of Unchanged Drug in Humans and Preclinical Animal Models: Increasing the Predictability of Poor Metabolism in Humans. Pharm Res. 2021 Jul; 38(7):1139-1156.
Bamfo NO, Hosey-Cojocari C, Benet LZ, Remsberg CM. PMID: 34254223; PMCID: PMC9855226.
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PubMed Mentions:
2 Fields:
Translation:
HumansAnimals
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Effects of Single Dose Rifampin on the Pharmacokinetics of Fluvastatin in Healthy Volunteers. Clin Pharmacol Ther. 2021 08; 110(2):480-485.
Xiang Y, Okochi H, Kozachenko I, Sodhi JK, Frassetto LA, Benet LZ. PMID: 33880760; PMCID: PMC9648157.
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PubMed Mentions:
2 Fields:
Translation:
Humans
-
There is Only One Valid Definition of Clearance: Critical Examination of Clearance Concepts Reveals the Potential for Errors in Clinical Drug Dosing Decisions. AAPS J. 2021 05 10; 23(3):67.
Benet LZ, Sodhi JK, Makrygiorgos G, Mesbah A. PMID: 33973074; PMCID: PMC8110503.
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PubMed Mentions:
7 Fields:
Translation:
Humans
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Tenofovir and emtricitabine concentrations in hair are comparable between individuals on tenofovir disoproxil fumarate versus tenofovir alafenamide-based ART. Drug Test Anal. 2021 Jul; 13(7):1354-1370.
Okochi H, Louie A, Phung N, Zhang K, Tallerico RM, Kuncze K, Spinelli MA, Koss CA, Benet LZ, Gandhi M. PMID: 33742745; PMCID: PMC9131373.
View in:
PubMed Mentions:
2 Translation:
Humans
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Investigating Intestinal Transporter Involvement in Rivaroxaban Disposition through Examination of Changes in Absorption. Pharm Res. 2021 May; 38(5):795-801.
Kou W, Sodhi JK, Wu X, Benet LZ. PMID: 33847849; PMCID: PMC8501891.
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PubMed Mentions:
4 Fields:
Translation:
HumansCells
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Using Individualized Patient Data for Prediction of Population Dosing Recommendations Versus Predictions of Individualized Patient Dosing. J Clin Pharmacol. 2021 06; 61(6):734-735.
Benet LZ. PMID: 33742720.
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PubMed Mentions: Fields:
Translation:
Humans
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Successful and Unsuccessful Prediction of Human Hepatic Clearance for Lead Optimization. J Med Chem. 2021 04 08; 64(7):3546-3559.
Sodhi JK, Benet LZ. PMID: 33765384; PMCID: PMC8504179.
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PubMed Mentions:
14 Fields:
Translation:
HumansCells
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Volume of Distribution is Unaffected by Metabolic Drug-Drug Interactions. Clin Pharmacokinet. 2021 02; 60(2):205-222.
Sodhi JK, Huang CH, Benet LZ. PMID: 32725383; PMCID: PMC7385331.
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PubMed Mentions:
4 Fields:
Translation:
Humans
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Intestinal Efflux Transporters P-gp and BCRP Are Not Clinically Relevant in Apixaban Disposition. Pharm Res. 2020 Sep 29; 37(10):208.
Sodhi JK, Liu S, Benet LZ. PMID: 32996065; PMCID: PMC7936879.
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PubMed Mentions:
7 Fields:
Translation:
Humans
-
Investigating the Theoretical Basis for In Vitro-In Vivo Extrapolation (IVIVE) in Predicting Drug Metabolic Clearance and Proposing Future Experimental Pathways. AAPS J. 2020 09 10; 22(5):120.
Benet LZ, Sodhi JK. PMID: 32914238; PMCID: PMC7515557.
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PubMed Mentions:
10 Fields:
Translation:
HumansAnimalsCells
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The Critical Role of Passive Permeability in Designing Successful Drugs. ChemMedChem. 2020 10 19; 15(20):1862-1874.
Di L, Artursson P, Avdeef A, Benet LZ, Houston JB, Kansy M, Kerns EH, Lennernäs H, Smith DA, Sugano K. PMID: 32743945.
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PubMed Mentions:
34 Fields:
Translation:
HumansAnimalsCells
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The Necessity of Using Changes in Absorption Time to Implicate Intestinal Transporter Involvement in Oral Drug-Drug Interactions. AAPS J. 2020 08 17; 22(5):111.
Sodhi JK, Benet LZ. PMID: 32808084; PMCID: PMC7478332.
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PubMed Mentions:
7 Fields:
Translation:
Humans
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A Simple Methodology to Differentiate Changes in Bioavailability From Changes in Clearance Following Oral Dosing of Metabolized Drugs. Clin Pharmacol Ther. 2020 08; 108(2):306-315.
Sodhi JK, Benet LZ. PMID: 32150643; PMCID: PMC7478330.
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PubMed Mentions:
7 Fields:
Translation:
Humans
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Are There Any Experimental Perfusion Data that Preferentially Support the Dispersion and Parallel-Tube Models over the Well-Stirred Model of Organ Elimination? Drug Metab Dispos. 2020 07; 48(7):537-543.
Sodhi JK, Wang HJ, Benet LZ. PMID: 32305951; PMCID: PMC7289046.
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PubMed Mentions:
13 Fields:
Translation:
Animals
-
Predicting Interactions between Rifampin and Antihypertensive Drugs Using the Biopharmaceutics Drug Disposition Classification System. Pharmacotherapy. 2020 04; 40(4):274-290.
Liu W, Yan T, Chen K, Yang L, Benet LZ, Zhai S. PMID: 32100890.
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PubMed Mentions:
4 Fields:
Translation:
Humans
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Challenging the Relevance of Unbound Tissue-to-Blood Partition Coefficient (Kpuu) on Prediction of Drug-Drug Interactions. Pharm Res. 2020 Mar 25; 37(4):73.
Sodhi JK, Liu S, Benet LZ. PMID: 32215750; PMCID: PMC7518636.
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PubMed Mentions:
4 Fields:
Translation:
Humans
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Late-Stage Failures of Monoclonal Antibody Drugs: A Retrospective Case Study Analysis. Pharmacology. 2020; 105(3-4):145-163.
Sun A, Benet LZ. PMID: 31910414.
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PubMed Mentions:
21 Fields:
Translation:
HumansAnimals
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Can BDDCS illuminate targets in drug design? Drug Discov Today. 2019 12; 24(12):2299-2306.
Bocci G, Benet LZ, Oprea TI. PMID: 31585170; PMCID: PMC7002033.
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PubMed Mentions:
3 Fields:
Translation:
HumansAnimals
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Protein Binding and Hepatic Clearance: Re-Examining the Discrimination between Models of Hepatic Clearance with Diazepam in the Isolated Perfused Rat Liver Preparation. Drug Metab Dispos. 2019 12; 47(12):1397-1402.
Wang HJ, Benet LZ. PMID: 31563869; PMCID: PMC7042717.
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PubMed Mentions:
3 Fields:
Translation:
AnimalsCells
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In Vitro-In Vivo Inaccuracy: The CYP3A4 Anomaly. Drug Metab Dispos. 2019 12; 47(12):1368-1371.
Bowman CM, Benet LZ. PMID: 31551322; PMCID: PMC7042718.
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PubMed Mentions:
5 Fields:
Translation:
HumansCells
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Food, Acid Supplementation and Drug Absorption - a Complicated Gastric Mix: a Randomized Control Trial. Pharm Res. 2019 Sep 04; 36(11):155.
Surofchy DD, Frassetto LA, Benet LZ. PMID: 31485804; PMCID: PMC7484952.
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PubMed Mentions:
1 Fields:
Translation:
Humans
-
How Transporters Have Changed Basic Pharmacokinetic Understanding. AAPS J. 2019 09 03; 21(6):103.
Benet LZ, Bowman CM, Sodhi JK. PMID: 31482335; PMCID: PMC7241423.
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PubMed Mentions:
13 Fields:
Translation:
HumansAnimals
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The Enhancement of Subcutaneous First-Pass Metabolism Causes Nonlinear Pharmacokinetics of TAK-448 after a Single Subcutaneous Administration to Rats. Drug Metab Dispos. 2019 09; 47(9):1004-1012.
Moriya Y, Kogame A, Tagawa Y, Morohashi A, Kondo T, Asahi S, Benet LZ. PMID: 31201213.
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PubMed Mentions:
1 Fields:
Translation:
HumansAnimals
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Interlaboratory Variability in Human Hepatocyte Intrinsic Clearance Values and Trends with Physicochemical Properties. Pharm Res. 2019 May 31; 36(8):113.
Bowman CM, Benet LZ. PMID: 31152241; PMCID: PMC7191673.
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PubMed Mentions:
7 Fields:
Translation:
HumansCells
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Understanding drug-drug interaction and pharmacogenomic changes in pharmacokinetics for metabolized drugs. J Pharmacokinet Pharmacodyn. 2019 04; 46(2):155-163.
Benet LZ, Bowman CM, Koleske ML, Rinaldi CL, Sodhi JK. PMID: 30911879; PMCID: PMC7179954.
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PubMed Mentions:
9 Fields:
Translation:
Humans
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In Vitro-In Vivo Extrapolation and Hepatic Clearance-Dependent Underprediction. J Pharm Sci. 2019 07; 108(7):2500-2504.
Bowman CM, Benet LZ. PMID: 30817922; PMCID: PMC7325626.
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PubMed Mentions:
17 Fields:
Translation:
HumansAnimalsCells
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Characterization of Fasiglifam-Related Liver Toxicity in Dogs. Drug Metab Dispos. 2019 05; 47(5):525-534.
Kogame A, Moriya Y, Mori I, Pan L, Morohashi A, Ebihara T, Fukui H, Tagawa Y, Benet LZ. PMID: 30765394.
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PubMed Mentions:
1 Fields:
Translation:
Animals
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The Presence of a Transporter-Induced Protein Binding Shift: A New Explanation for Protein-Facilitated Uptake and Improvement for In Vitro-In Vivo Extrapolation. Drug Metab Dispos. 2019 04; 47(4):358-363.
Bowman CM, Okochi H, Benet LZ. PMID: 30674616; PMCID: PMC6413769.
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PubMed Mentions:
13 Fields:
Translation:
AnimalsCells
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Evaluating Within-Subject Variability for Narrow Therapeutic Index Drugs. Clin Pharmacol Ther. 2019 02; 105(2):411-416.
Jayachandran P, Okochi H, Frassetto LA, Park W, Fang L, Zhao L, Benet LZ. PMID: 30652304.
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PubMed Mentions:
4 Fields:
Translation:
HumansCTClinical Trials
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Batch-to-Batch and Within-Subject Variability: What Do We Know and How Do These Variabilities Affect Clinical Pharmacology and Bioequivalence? Clin Pharmacol Ther. 2019 02; 105(2):326-328.
Benet LZ, Jayachandran P, Carroll KJ, Burmeister Getz E. PMID: 30652313.
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PubMed Mentions:
3 Fields:
Translation:
Humans
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TPT sulfonate, a single, oral dose schistosomicidal prodrug: In vivo efficacy, disposition and metabolic profiling. Int J Parasitol Drugs Drug Resist. 2018 12; 8(3):571-586.
Wolfe AR, Neitz RJ, Burlingame M, Suzuki BM, Lim KC, Scheideler M, Nelson DL, Benet LZ, Caffrey CR. PMID: 30503203; PMCID: PMC6287543.
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PubMed Mentions:
7 Fields:
Translation:
Animals
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The Extended Clearance Concept Following Oral and Intravenous Dosing: Theory and Critical Analyses. Pharm Res. 2018 Oct 22; 35(12):242.
Benet LZ, Bowman CM, Liu S, Sodhi JK. PMID: 30349948; PMCID: PMC6364828.
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PubMed Mentions:
14 Fields:
Translation:
HumansCells
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Ascorbic acid metabolites are involved in intraocular pressure control in the general population. Redox Biol. 2019 01; 20:349-353.
Hysi PG, Khawaja AP, Menni C, Tamraz B, Wareham N, Khaw KT, Foster PJ, Benet LZ, Spector TD, Hammond CJ. PMID: 30391827; PMCID: PMC6223183.
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PubMed Mentions:
23 Fields:
Translation:
HumansPHPublic Health
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Development and Validation of an Immunoassay for Tenofovir in Urine as a Real-Time Metric of Antiretroviral Adherence. EClinicalMedicine. 2018 Aug-Sep; 2-3:22-28.
Gandhi M, Bacchetti P, Rodrigues WC, Spinelli M, Koss CA, Drain PK, Baeten JM, Mugo NR, Ngure K, Benet LZ, Okochi H, Wang G, Vincent M. PMID: 30906930; PMCID: PMC6428441.
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PubMed Mentions:
42
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An examination of protein binding and protein-facilitated uptake relating to in vitro-in vivo extrapolation. Eur J Pharm Sci. 2018 Oct 15; 123:502-514.
Bowman CM, Benet LZ. PMID: 30098391; PMCID: PMC6365006.
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PubMed Mentions:
23 Fields:
Translation:
HumansAnimalsCells
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Evaluation of the Relevance of DILI Predictive Hypotheses in Early Drug Development: Review of In Vitro Methodologies vs BDDCS Classification. Toxicol Res (Camb). 2018 May 08; 7(3):358-370.
Chan R, Benet LZ. PMID: 29785262; PMCID: PMC5959290.
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PubMed Mentions:
4
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Predicting Pharmacokinetics/Pharmacodynamics in the Individual Patient: Separating Reality From Hype. J Clin Pharmacol. 2018 Aug; 58(8):979-989.
Benet LZ. PMID: 29663413.
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PubMed Mentions:
2 Fields:
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Measures of BSEP Inhibition In Vitro Are Not Useful Predictors of DILI. Toxicol Sci. 2018 04 01; 162(2):499-508.
Chan R, Benet LZ. PMID: 29272540; PMCID: PMC5888978.
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PubMed Mentions:
20 Fields:
Translation:
HumansAnimalsCells
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A Drug-drug Interaction Between Cyclosporine and Nystatin. Clin Ther. 2018 04; 40(4):660-662.
Liu W, Guan X, Yu Z, Chen K, Benet L, Zhai S. PMID: 29551534.
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PubMed Mentions:
3 Fields:
Translation:
Humans
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Development and validation of an assay to analyze atazanavir in human hair via liquid chromatography/tandem mass spectrometry. Rapid Commun Mass Spectrom. 2018 Mar 15; 32(5):431-441.
Phung N, Kuncze K, Okochi H, Louie A, Benet LZ, Ofokotun I, Haas DW, Currier JS, Chawana TD, Sheth AN, Bacchetti P, Gandhi M, Horng H. PMID: 29315954; PMCID: PMC5848502.
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PubMed Mentions:
8 Fields:
Translation:
Humans
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Why Drugs Fail in Late Stages of Development: Case Study Analyses from the Last Decade and Recommendations. AAPS J. 2018 03 13; 20(3):46.
Parasrampuria DA, Benet LZ, Sharma A. PMID: 29536211.
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PubMed Mentions:
25 Fields:
Translation:
Humans
-
View in:
PubMed Mentions:
2 Fields:
Translation:
HumansAnimalsCells
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Comparison of Measures of Adherence to Human Immunodeficiency Virus Preexposure Prophylaxis Among Adolescent and Young Men Who Have Sex With Men in the United States. Clin Infect Dis. 2018 01 06; 66(2):213-219.
Koss CA, Hosek SG, Bacchetti P, Anderson PL, Liu AY, Horng H, Benet LZ, Kuncze K, Louie A, Saberi P, Wilson CM, Gandhi M. PMID: 29020194; PMCID: PMC5850042.
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PubMed Mentions:
64 Fields:
Translation:
HumansPHPublic Health
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The Universally Unrecognized Assumption in Predicting Drug Clearance and Organ Extraction Ratio. Clin Pharmacol Ther. 2018 03; 103(3):521-525.
Benet LZ, Liu S, Wolfe AR. PMID: 28762489; PMCID: PMC6364827.
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PubMed Mentions:
14 Fields:
Translation:
Humans
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Commentary on: "Influence of OATP1B1 Function on the Disposition of Sorafenib-β-D-Glucuronide". Clin Transl Sci. 2017 07; 10(4):240-241.
Morrissey KM, Benet LZ, Ware JA. PMID: 28664655; PMCID: PMC5504478.
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PubMed Mentions:
1 Fields:
Translation:
Cells
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Understanding the Potential Interethnic Difference in Rosuvastatin Pharmacokinetics. J Pharm Sci. 2017 09; 106(9):2231-2233.
Benet LZ, Wu HF. PMID: 28502797.
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PubMed Mentions:
1 Fields:
Translation:
Humans
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Cellular Uptake of Levocetirizine by Organic Anion Transporter 4. J Pharm Sci. 2017 09; 106(9):2895-2898.
Noguchi S, Nishimura T, Mukaida S, Benet LZ, Nakashima E, Tomi M. PMID: 28385546.
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PubMed Mentions:
6 Fields:
Translation:
HumansCells
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Rosuvastatin Pharmacokinetics in Asian and White Subjects Wild Type for Both OATP1B1 and BCRP Under Control and Inhibited Conditions. J Pharm Sci. 2017 09; 106(9):2751-2757.
Wu HF, Hristeva N, Chang J, Liang X, Li R, Frassetto L, Benet LZ. PMID: 28385543; PMCID: PMC5675025.
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PubMed Mentions:
32 Fields:
Translation:
HumansCTClinical Trials
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Evaluation of DILI Predictive Hypotheses in Early Drug Development. Chem Res Toxicol. 2017 04 17; 30(4):1017-1029.
Chan R, Benet LZ. PMID: 28257576; PMCID: PMC5674994.
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PubMed Mentions:
10 Fields:
Translation:
Humans
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Differences in Cumulative Exposure and Adherence to Tenofovir in the VOICE, iPrEx OLE, and PrEP Demo Studies as Determined via Hair Concentrations. AIDS Res Hum Retroviruses. 2017 08; 33(8):778-783.
Koss CA, Bacchetti P, Hillier SL, Livant E, Horng H, Mgodi N, Mirembe BG, Gomez Feliciano K, Horn S, Liu AY, Glidden DV, Grant RM, Benet LZ, Louie A, van der Straten A, Chirenje ZM, Marrazzo JM, Gandhi M. PMID: 28253024; PMCID: PMC5564054.
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PubMed Mentions:
45 Fields:
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Meal Effects Confound Attempts to Counteract Rabeprazole-Induced Hypochlorhydria Decreases in Atazanavir Absorption. Pharm Res. 2017 03; 34(3):619-628.
Faber KP, Wu HF, Yago MR, Xu X, Kadiyala P, Frassetto LA, Benet LZ. PMID: 28028768; PMCID: PMC7179955.
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PubMed Mentions:
6 Fields:
Translation:
Humans
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Classification of natural products as sources of drugs according to the biopharmaceutics drug disposition classification system (BDDCS). Chin J Nat Med. 2016 Dec; 14(12):888-897.
Li J, Larregieu CA, Benet LZ. PMID: 28262115.
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PubMed Mentions:
12 Fields:
Translation:
HumansAnimals
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Between-Batch Pharmacokinetic Variability Inflates Type I Error Rate in Conventional Bioequivalence Trials: A Randomized Advair Diskus Clinical Trial. Clin Pharmacol Ther. 2017 03; 101(3):331-340.
Burmeister Getz E, Carroll KJ, Mielke J, Benet LZ, Jones B. PMID: 27727445; PMCID: PMC5324827.
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PubMed Mentions:
7 Fields:
Translation:
Humans
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Association of age, baseline kidney function, and medication exposure with declines in creatinine clearance on pre-exposure prophylaxis: an observational cohort study. Lancet HIV. 2016 11; 3(11):e521-e528.
Gandhi M, Glidden DV, Mayer K, Schechter M, Buchbinder S, Grinsztejn B, Hosek S, Casapia M, Guanira J, Bekker LG, Louie A, Horng H, Benet LZ, Liu A, Grant RM. PMID: 27658870; PMCID: PMC5085869.
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Hepatic Clearance Predictions from In Vitro-In Vivo Extrapolation and the Biopharmaceutics Drug Disposition Classification System. Drug Metab Dispos. 2016 11; 44(11):1731-1735.
Bowman CM, Benet LZ. PMID: 27519549; PMCID: PMC11024986.
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PubMed Mentions:
20 Fields:
Translation:
HumansCells
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2016 Remington Honor Medal Address: Science for the profession. J Am Pharm Assoc (2003). 2016 Jul-Aug; 56(4):365-8.
Benet LZ. PMID: 27450136.
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PubMed Mentions: Fields:
Translation:
Humans
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Isoniazid hair concentrations in children with tuberculosis: a proof of concept study. Int J Tuberc Lung Dis. 2016 06; 20(6):844-7.
Mave V, Chandanwale A, Kinikar A, Khadse S, Kagal A, Gupte N, Suryavanshi N, Nimkar S, Koli H, Khwaja S, Bharadwaj R, Joshi S, Horng H, Benet LZ, Ramachandran G, Dooley KE, Gupta A, Gandhi M. PMID: 27155191; PMCID: PMC4889729.
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PubMed Mentions:
5 Fields:
Translation:
Humans
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BDDCS, the Rule of 5 and drugability. Adv Drug Deliv Rev. 2016 06 01; 101:89-98.
Benet LZ, Hosey CM, Ursu O, Oprea TI. PMID: 27182629; PMCID: PMC4910824.
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PubMed Mentions:
224 Fields:
Translation:
HumansAnimals
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Batch-to-batch pharmacokinetic variability confounds current bioequivalence regulations: A dry powder inhaler randomized clinical trial. Clin Pharmacol Ther. 2016 Sep; 100(3):223-31.
Burmeister Getz E, Carroll KJ, Jones B, Benet LZ. PMID: 27037630; PMCID: PMC5102576.
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PubMed Mentions:
14 Fields:
Translation:
Humans
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Use of the Biopharmaceutics Drug Disposition Classification System (BDDCS) to Help Predict the Occurrence of Idiosyncratic Cutaneous Adverse Drug Reactions Associated with Antiepileptic Drug Usage. AAPS J. 2016 05; 18(3):757-66.
Chan R, Wei CY, Chen YT, Benet LZ. PMID: 26951484; PMCID: PMC5256615.
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PubMed Mentions:
6 Fields:
Translation:
Humans
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Reliability of In Vitro and In Vivo Methods for Predicting the Effect of P-Glycoprotein on the Delivery of Antidepressants to the Brain. Clin Pharmacokinet. 2016 Feb; 55(2):143-67.
Zheng Y, Chen X, Benet LZ. PMID: 26293617; PMCID: PMC5674979.
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PubMed Mentions:
9 Fields:
Translation:
HumansAnimals
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BDDCS Predictions, Self-Correcting Aspects of BDDCS Assignments, BDDCS Assignment Corrections, and Classification for more than 175 Additional Drugs. AAPS J. 2016 Jan; 18(1):251-60.
Hosey CM, Chan R, Benet LZ. PMID: 26589308; PMCID: PMC4706282.
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PubMed Mentions:
30 Fields:
Translation:
Humans
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Few Drugs Display Flip-Flop Pharmacokinetics and These Are Primarily Associated with Classes 3 and 4 of the BDDCS. J Pharm Sci. 2015 Sep; 104(9):3229-35.
Garrison KL, Sahin S, Benet LZ. PMID: 26010239; PMCID: PMC4536115.
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PubMed Mentions:
14 Fields:
Translation:
HumansAnimals
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Predicting the extent of metabolism using in vitro permeability rate measurements and in silico permeability rate predictions. Mol Pharm. 2015 May 04; 12(5):1456-66.
Hosey CM, Benet LZ. PMID: 25816851; PMCID: PMC4666302.
View in:
PubMed Mentions:
15 Fields:
Translation:
HumansAnimalsCells
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pH Dependent but not P-gp Dependent Bidirectional Transport Study of S-propranolol: The Importance of Passive Diffusion. Pharm Res. 2015 Aug; 32(8):2516-26.
Zheng Y, Benet LZ, Okochi H, Chen X. PMID: 25690341; PMCID: PMC4891189.
View in:
PubMed Mentions:
9 Fields:
Translation:
HumansAnimalsCells
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A phase I study of targeted, dose-escalated intravenous busulfan in combination with etoposide as myeloablative therapy for autologous stem cell transplantation in acute myeloid leukemia. Clin Lymphoma Myeloma Leuk. 2015 Jun; 15(6):377-83.
Mannis GN, Andreadis C, Logan AC, Damon LE, Benet LZ, Ai WZ, Gaensler KM, Kaplan LD, Koplowicz YB, Linker CA, Olin RL, Sayre PH, Smith CC, Sudhindra A, Venstrom JM, Wolf JL, Martin TG. PMID: 25776193.
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PubMed Mentions:
1 Fields:
Translation:
HumansCTClinical Trials
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Inclusion of placebos and blinding for ascending dose first-in-human studies and other underpowered phase 1 studies has not been justified and on balance is not useful. Basic Clin Pharmacol Toxicol. 2015 Jul; 117(1):44-51.
Parasrampuria DA, Benet LZ. PMID: 25406995.
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PubMed Mentions:
7 Fields:
Translation:
Humans
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The use of betaine HCl to enhance dasatinib absorption in healthy volunteers with rabeprazole-induced hypochlorhydria. AAPS J. 2014 Nov; 16(6):1358-65.
Yago MR, Frymoyer A, Benet LZ, Smelick GS, Frassetto LA, Ding X, Dean B, Salphati L, Budha N, Jin JY, Dresser MJ, Ware JA. PMID: 25274610; PMCID: PMC4389759.
View in:
PubMed Mentions:
13 Fields:
Translation:
Humans
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Predicting when biliary excretion of parent drug is a major route of elimination in humans. AAPS J. 2014 Sep; 16(5):1085-96.
Hosey CM, Broccatelli F, Benet LZ. PMID: 25004821; PMCID: PMC4147063.
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PubMed Mentions:
9 Fields:
Translation:
Humans
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Distinguishing between the permeability relationships with absorption and metabolism to improve BCS and BDDCS predictions in early drug discovery. Mol Pharm. 2014 Apr 07; 11(4):1335-44.
Larregieu CA, Benet LZ. PMID: 24628254; PMCID: PMC3983369.
View in:
PubMed Mentions:
12 Fields:
Translation:
HumansCells
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Best single time point correlations with AUC for cyclosporine and tacrolimus in HIV-infected kidney and liver transplant recipients. Transplantation. 2014 Mar 27; 97(6):702-7.
Frassetto LA, Tan-Tam CC, Barin B, Browne M, Wolfe AR, Stock PG, Roland M, Benet LZ. PMID: 24389906; PMCID: PMC4018220.
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PubMed Mentions:
5 Fields:
Translation:
Humans
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Mouse liver repopulation with hepatocytes generated from human fibroblasts. Nature. 2014 Apr 03; 508(7494):93-7.
Zhu S, Rezvani M, Harbell J, Mattis AN, Wolfe AR, Benet LZ, Willenbring H, Ding S. PMID: 24572354; PMCID: PMC4161230.
View in:
PubMed Mentions:
136 Fields:
Translation:
HumansAnimalsCells
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Prevalence of acid-reducing agents (ARA) in cancer populations and ARA drug-drug interaction potential for molecular targeted agents in clinical development. Mol Pharm. 2013 Nov 04; 10(11):4055-62.
Smelick GS, Heffron TP, Chu L, Dean B, West DA, Duvall SL, Lum BL, Budha N, Holden SN, Benet LZ, Frymoyer A, Dresser MJ, Ware JA. PMID: 24044612.
View in:
PubMed Mentions:
59 Fields:
Translation:
Humans
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Effect of P-glycoprotein on the rat intestinal permeability and metabolism of the BDDCS class 1 drug verapamil. Mol Pharm. 2013 Nov 04; 10(11):4038-45.
Estudante M, Maya M, Morais JG, Soveral G, Benet LZ. PMID: 24044638.
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PubMed Mentions: Fields:
Translation:
Animals
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Changes in clearance, volume and bioavailability of immunosuppressants when given with HAART in HIV-1 infected liver and kidney transplant recipients. Biopharm Drug Dispos. 2013 Nov; 34(8):442-51.
Frassetto L, Floren L, Barin B, Browne M, Wolfe A, Roland M, Stock P, Carlson L, Christians U, Benet L. PMID: 24030928; PMCID: PMC4018225.
View in:
PubMed Mentions:
11 Fields:
Translation:
HumansCellsCTClinical Trials
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Gastric reacidification with betaine HCl in healthy volunteers with rabeprazole-induced hypochlorhydria. Mol Pharm. 2013 Nov 04; 10(11):4032-7.
Yago MR, Frymoyer AR, Smelick GS, Frassetto LA, Budha NR, Dresser MJ, Ware JA, Benet LZ. PMID: 23980906; PMCID: PMC3946491.
View in:
PubMed Mentions:
7 Fields:
Translation:
HumansCTClinical Trials
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The nonenzymatic reactivity of the acyl-linked metabolites of mefenamic acid toward amino and thiol functional group bionucleophiles. Drug Metab Dispos. 2013 Nov; 41(11):1923-33.
Horng H, Benet LZ. PMID: 23975029; PMCID: PMC3807055.
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PubMed Mentions:
2 Fields:
Translation:
AnimalsCells
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Characterization of the acyl-adenylate linked metabolite of mefenamic Acid. Chem Res Toxicol. 2013 Mar 18; 26(3):465-76.
Horng H, Benet LZ. PMID: 23402341; PMCID: PMC3626286.
View in:
PubMed Mentions:
1 Fields:
Translation:
AnimalsCells
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Pharmacokinetics and metabolism of 2-aminothiazoles with antiprion activity in mice. Pharm Res. 2013 Apr; 30(4):932-50.
Silber BM, Rao S, Fife KL, Gallardo-Godoy A, Renslo AR, Dalvie DK, Giles K, Freyman Y, Elepano M, Gever JR, Li Z, Jacobson MP, Huang Y, Benet LZ, Prusiner SB. PMID: 23417511; PMCID: PMC3640342.
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PubMed Mentions:
16 Fields:
Translation:
HumansAnimalsCells
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Drug discovery and regulatory considerations for improving in silico and in vitro predictions that use Caco-2 as a surrogate for human intestinal permeability measurements. AAPS J. 2013 Apr; 15(2):483-97.
Larregieu CA, Benet LZ. PMID: 23344793; PMCID: PMC3675726.
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PubMed Mentions:
46 Fields:
Translation:
HumansCells
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The role of BCS (biopharmaceutics classification system) and BDDCS (biopharmaceutics drug disposition classification system) in drug development. J Pharm Sci. 2013 Jan; 102(1):34-42.
Benet LZ. PMID: 23147500; PMCID: PMC3684558.
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PubMed Mentions:
67 Fields:
Translation:
HumansAnimalsCells
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A step closer to personalized chemotherapy: consideration of the influence of genetic variation in hepatic uptake transporters on the metabolism of CYP3A substrates. Clin Pharmacol Ther. 2012 Nov; 92(5):551-2.
Benet LZ. PMID: 23085879.
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PubMed Mentions: Fields:
Translation:
HumansAnimals
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Intestinal drug transporters: an overview. Adv Drug Deliv Rev. 2013 Oct; 65(10):1340-56.
Estudante M, Morais JG, Soveral G, Benet LZ. PMID: 23041352.
View in:
PubMed Mentions:
79 Fields:
Translation:
HumansAnimals
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Drug absorption interactions between oral targeted anticancer agents and PPIs: is pH-dependent solubility the Achilles heel of targeted therapy? Clin Pharmacol Ther. 2012 Aug; 92(2):203-13.
Budha NR, Frymoyer A, Smelick GS, Jin JY, Yago MR, Dresser MJ, Holden SN, Benet LZ, Ware JA. PMID: 22739140.
View in:
PubMed Mentions:
94 Fields:
Translation:
Humans
-
Benet L Z and Galeazzi R L: noncompartmental determination of the steady-state volume of distribution, J Pharm Sci 68, 1071-1074, 1979--the backstory. AAPS J. 2012 Jun; 14(2):164-7.
Benet LZ. PMID: 22302585; PMCID: PMC3326156.
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PubMed Mentions:
4 Fields:
Translation:
HumansAnimals
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Sotalol permeability in cultured-cell, rat intestine, and PAMPA system. Pharm Res. 2012 Jul; 29(7):1768-74.
Liu W, Okochi H, Benet LZ, Zhai SD. PMID: 22350803; PMCID: PMC4167886.
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PubMed Mentions:
6 Fields:
Translation:
AnimalsCells
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BDDCS class prediction for new molecular entities. Mol Pharm. 2012 Mar 05; 9(3):570-80.
Broccatelli F, Cruciani G, Benet LZ, Oprea TI. PMID: 22224483; PMCID: PMC3295927.
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PubMed Mentions:
22 Fields:
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Improving the prediction of the brain disposition for orally administered drugs using BDDCS. Adv Drug Deliv Rev. 2012 Jan; 64(1):95-109.
Broccatelli F, Larregieu CA, Cruciani G, Oprea TI, Benet LZ. PMID: 22261306; PMCID: PMC3496430.
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PubMed Mentions:
22 Fields:
Translation:
HumansAnimals
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Impact of a hospitalwide increase in empiric pediatric vancomycin dosing on initial trough concentrations. Pharmacotherapy. 2011 Sep; 31(9):871-6.
Frymoyer A, Guglielmo BJ, Wilson SD, Scarpace SB, Benet LZ, Hersh AL. PMID: 21923588; PMCID: PMC3727161.
View in:
PubMed Mentions:
18 Fields:
Translation:
HumansCells
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Pharmacokinetic differences corroborate observed low tacrolimus dosage in Native American renal transplant patients. Drug Metab Dispos. 2011 Nov; 39(11):2017-9.
Grover A, Frassetto LA, Benet LZ, Chakkera HA. PMID: 21849516; PMCID: PMC3198899.
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PubMed Mentions:
14 Fields:
Translation:
Humans
-
BDDCS applied to over 900 drugs. AAPS J. 2011 Dec; 13(4):519-47.
Benet LZ, Broccatelli F, Oprea TI. PMID: 21818695; PMCID: PMC3231854.
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PubMed Mentions:
172 Fields:
Translation:
Cells
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Lead PK commentary: predicting human pharmacokinetics. J Pharm Sci. 2011 Oct; 100(10):4047-9.
Rowland M, Benet LZ. PMID: 21630278.
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PubMed Mentions:
12 Fields:
Translation:
HumansAnimals
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Professor Akira Tsuji: scientist, educator, and leader. J Pharm Sci. 2011 Sep; 100(9):3541-6.
Terasaki T, Sugiyama Y, Benet LZ. PMID: 21630279.
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PubMed Mentions: Fields:
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Effects of uremic toxins on transport and metabolism of different biopharmaceutics drug disposition classification system xenobiotics. J Pharm Sci. 2011 Sep; 100(9):3831-42.
Reyes M, Benet LZ. PMID: 21618544; PMCID: PMC3581075.
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PubMed Mentions:
19 Fields:
Translation:
HumansAnimalsCells
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Intermittent drug dosing intervals guided by the operational multiple dosing half lives for predictable plasma accumulation and fluctuation. J Pharmacokinet Pharmacodyn. 2011 Jun; 38(3):369-83.
Grover A, Benet LZ. PMID: 21499748; PMCID: PMC3677834.
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PubMed Mentions:
5 Fields:
Translation:
HumansCells
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The BCS, BDDCS, and regulatory guidances. Pharm Res. 2011 Jul; 28(7):1774-8.
Chen ML, Amidon GL, Benet LZ, Lennernas H, Yu LX. PMID: 21491148.
View in:
PubMed Mentions:
21 Fields:
Translation:
Humans
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Is Ciprofloxacin a Substrate of P-glycoprotein? Arch Drug Inf. 2011 Mar; 4(1):1-9.
Park MS, Okochi H, Benet LZ. PMID: 21572514; PMCID: PMC3084506.
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PubMed Mentions:
13
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Founding figures of pharmacokinetics: tribute to Malcolm Rowland. J Pharmacokinet Pharmacodyn. 2010 Dec; 37(6):525-7.
Aarons L, Benet LZ. PMID: 21069561.
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PubMed Mentions: Fields:
Translation:
HumansAnimals
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Clearance (née Rowland) concepts: a downdate and an update. J Pharmacokinet Pharmacodyn. 2010 Dec; 37(6):529-39.
Benet LZ. PMID: 21113650; PMCID: PMC3005114.
View in:
PubMed Mentions:
8 Fields:
Translation:
HumansAnimals
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Age and sex differences in the effects of the immunosuppressants cyclosporine, sirolimus and everolimus on rat brain metabolism. Neurotoxicology. 2011 Jan; 32(1):50-7.
Gottschalk S, Cummins CL, Leibfritz D, Christians U, Benet LZ, Serkova NJ. PMID: 21075140.
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PubMed Mentions:
19 Fields:
Translation:
Animals
-
Effect of single-dose rifampin on the pharmacokinetics of warfarin in healthy volunteers. Clin Pharmacol Ther. 2010 Oct; 88(4):540-7.
Frymoyer A, Shugarts S, Browne M, Wu AH, Frassetto L, Benet LZ. PMID: 20703222; PMCID: PMC3091944.
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PubMed Mentions:
13 Fields:
Translation:
HumansAnimals
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The FDA should eliminate the ambiguities in the current BCS biowaiver guidance and make public the drugs for which BCS biowaivers have been granted. Clin Pharmacol Ther. 2010 Sep; 88(3):405-7.
Benet LZ, Larregieu CA. PMID: 20668447; PMCID: PMC4169211.
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PubMed Mentions:
11 Fields:
Translation:
HumansAnimals
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Prediction of vancomycin pharmacodynamics in children with invasive methicillin-resistant Staphylococcus aureus infections: a Monte Carlo simulation. Clin Ther. 2010 Mar; 32(3):534-42.
Frymoyer A, Hersh AL, Coralic Z, Benet LZ, Joseph Guglielmo B. PMID: 20399990; PMCID: PMC3097025.
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PubMed Mentions:
21 Fields:
Translation:
HumansCells
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Membrane transporters in drug development. Nat Rev Drug Discov. 2010 Mar; 9(3):215-36.
International Transporter Consortium, Giacomini KM, Huang SM, Tweedie DJ, Benet LZ, Brouwer KL, Chu X, Dahlin A, Evers R, Fischer V, Hillgren KM, Hoffmaster KA, Ishikawa T, Keppler D, Kim RB, Lee CA, Niemi M, Polli JW, Sugiyama Y, Swaan PW, Ware JA, Wright SH, Yee SW, Zamek-Gliszczynski MJ, Zhang L. PMID: 20190787; PMCID: PMC3326076.
View in:
PubMed Mentions:
1030 Fields:
Translation:
HumansAnimals
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Hepatic clearance, but not gut availability, of erythromycin is altered in patients with end-stage renal disease. Clin Pharmacol Ther. 2010 Apr; 87(4):465-72.
Sun H, Frassetto LA, Huang Y, Benet LZ. PMID: 20090676; PMCID: PMC3581054.
View in:
PubMed Mentions:
18 Fields:
Translation:
Humans
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Stereoselective flunoxaprofen-S-acyl-glutathione thioester formation mediated by acyl-CoA formation in rat hepatocytes. Drug Metab Dispos. 2010 Jan; 38(1):133-42.
Grillo MP, Wait JC, Tadano Lohr M, Khera S, Benet LZ. PMID: 19786506; PMCID: PMC2802421.
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PubMed Mentions:
2 Fields:
Translation:
AnimalsCells
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Predicting drug disposition via application of a Biopharmaceutics Drug Disposition Classification System. Basic Clin Pharmacol Toxicol. 2010 Mar; 106(3):162-7.
Benet LZ. PMID: 20002064; PMCID: PMC3564954.
View in:
PubMed Mentions:
30 Fields:
Translation:
Humans
-
The drug transporter-metabolism alliance: uncovering and defining the interplay. Mol Pharm. 2009 Nov-Dec; 6(6):1631-43.
Benet LZ. PMID: 19874004; PMCID: PMC2796475.
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PubMed Mentions:
51 Fields:
Translation:
HumansAnimalsCells
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Comparison of bidirectional lamivudine and zidovudine transport using MDCK, MDCK-MDR1, and Caco-2 cell monolayers. J Pharm Sci. 2009 Nov; 98(11):4413-9.
de Souza J, Benet LZ, Huang Y, Storpirtis S. PMID: 19472342.
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PubMed Mentions:
22 Fields:
Translation:
HumansAnimalsCells
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A Holy Grail of clinical pharmacology: prediction of drug pharmacokinetics and pharmacodynamics in the individual patient. Clin Pharmacol Ther. 2009 Aug; 86(2):133-4.
Benet LZ. PMID: 19621007.
View in:
PubMed Mentions:
1 Fields:
Translation:
HumansCells
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The role of transporters in the pharmacokinetics of orally administered drugs. Pharm Res. 2009 Sep; 26(9):2039-54.
Shugarts S, Benet LZ. PMID: 19568696; PMCID: PMC2719753.
View in:
PubMed Mentions:
131 Fields:
Translation:
HumansAnimals
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Current recommended dosing of vancomycin for children with invasive methicillin-resistant Staphylococcus aureus infections is inadequate. Pediatr Infect Dis J. 2009 May; 28(5):398-402.
Frymoyer A, Hersh AL, Benet LZ, Guglielmo BJ. PMID: 19295465; PMCID: PMC3101254.
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PubMed Mentions:
49 Fields:
Translation:
HumansCells
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Effects of drug transporters on volume of distribution. AAPS J. 2009 Jun; 11(2):250-61.
Grover A, Benet LZ. PMID: 19399628; PMCID: PMC2691462.
View in:
PubMed Mentions:
46 Fields:
Translation:
HumansAnimals
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Nonnucleoside reverse transcriptase inhibitor pharmacokinetics in a large unselected cohort of HIV-infected women. J Acquir Immune Defic Syndr. 2009 Apr 15; 50(5):482-91.
Gandhi M, Benet LZ, Bacchetti P, Kalinowski A, Anastos K, Wolfe AR, Young M, Cohen M, Minkoff H, Gange SJ, Greenblatt RM, Women's Interagency HIV Study. PMID: 19408353; PMCID: PMC2700138.
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PubMed Mentions:
16 Fields:
Translation:
Humans
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The operational multiple dosing half-life: a key to defining drug accumulation in patients and to designing extended release dosage forms. Pharm Res. 2008 Dec; 25(12):2869-77.
Sahin S, Benet LZ. PMID: 19015955; PMCID: PMC3581066.
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PubMed Mentions:
41 Fields:
Translation:
Humans
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Elucidating rifampin's inducing and inhibiting effects on glyburide pharmacokinetics and blood glucose in healthy volunteers: unmasking the differential effects of enzyme induction and transporter inhibition for a drug and its primary metabolite. Clin Pharmacol Ther. 2009 Jan; 85(1):78-85.
Zheng HX, Huang Y, Frassetto LA, Benet LZ. PMID: 18843263; PMCID: PMC3582657.
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PubMed Mentions:
46 Fields:
Translation:
HumansCTClinical Trials
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Moringa oleifera leaf extracts inhibit 6beta-hydroxylation of testosterone by CYP3A4. J Infect Dev Ctries. 2008 Oct 01; 2(5):379-83.
Monera TG, Wolfe AR, Maponga CC, Benet LZ, Guglielmo J. PMID: 19745507; PMCID: PMC5385924.
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PubMed Mentions:
15 Fields:
Translation:
HumansAnimalsCells
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Gamma-glutamyltranspeptidase-mediated degradation of diclofenac-S-acyl-glutathione in vitro and in vivo in rat. Chem Res Toxicol. 2008 Oct; 21(10):1933-8.
Grillo MP, Hua F, March KL, Benet LZ, Knutson CG, Ware JA. PMID: 18693772.
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PubMed Mentions:
2 Fields:
Translation:
AnimalsCells
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The use of BDDCS in classifying the permeability of marketed drugs. Pharm Res. 2008 Mar; 25(3):483-8.
Benet LZ, Amidon GL, Barends DM, Lennernäs H, Polli JE, Shah VP, Stavchansky SA, Yu LX. PMID: 18236138; PMCID: PMC3580995.
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PubMed Mentions:
29 Fields:
Translation:
Humans
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Differential effects of fibrates on the metabolic activation of 2-phenylpropionic acid in rats. Drug Metab Dispos. 2008 Apr; 36(4):682-7.
Li C, Grillo MP, Badagnani I, Fife KL, Benet LZ. PMID: 18187563.
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PubMed Mentions: Fields:
Translation:
AnimalsCells
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HIV-infected liver and kidney transplant recipients: 1- and 3-year outcomes. Am J Transplant. 2008 Feb; 8(2):355-65.
Roland ME, Barin B, Carlson L, Frassetto LA, Terrault NA, Hirose R, Freise CE, Benet LZ, Ascher NL, Roberts JP, Murphy B, Keller MJ, Olthoff KM, Blumberg EA, Brayman KL, Bartlett ST, Davis CE, McCune JM, Bredt BM, Stablein DM, Stock PG. PMID: 18093266.
View in:
PubMed Mentions:
79 Fields:
Translation:
Humans
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Predicting drug disposition, absorption/elimination/transporter interplay and the role of food on drug absorption. Adv Drug Deliv Rev. 2008 Mar 17; 60(6):717-33.
Custodio JM, Wu CY, Benet LZ. PMID: 18199522; PMCID: PMC2292816.
View in:
PubMed Mentions:
99 Fields:
Translation:
Humans
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Immunosuppressant pharmacokinetics and dosing modifications in HIV-1 infected liver and kidney transplant recipients. Am J Transplant. 2007 Dec; 7(12):2816-20.
Frassetto LA, Browne M, Cheng A, Wolfe AR, Roland ME, Stock PG, Carlson L, Benet LZ. PMID: 17949460.
View in:
PubMed Mentions:
43 Fields:
Translation:
HumansCellsCTClinical Trials
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Assessment and validation of the MS/MS fragmentation patterns of the macrolide immunosuppressant everolimus. J Mass Spectrom. 2007 Jun; 42(6):793-802.
Boernsen KO, Egge-Jacobsen W, Inverardi B, Strom T, Streit F, Schiebel HM, Benet LZ, Christians U. PMID: 17511017.
View in:
PubMed Mentions:
8 Fields:
Translation:
Cells
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Effects of uptake and efflux transporter inhibition on erythromycin breath test results. Clin Pharmacol Ther. 2007 Jun; 81(6):828-32.
Frassetto LA, Poon S, Tsourounis C, Valera C, Benet LZ. PMID: 17361125.
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PubMed Mentions:
19 Fields:
Translation:
Humans
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Studies on the metabolism of tolmetin to the chemically reactive acyl-coenzyme A thioester intermediate in rats. Drug Metab Dispos. 2007 May; 35(5):758-64.
Olsen J, Li C, Skonberg C, Bjørnsdottir I, Sidenius U, Benet LZ, Hansen SH. PMID: 17303625.
View in:
PubMed Mentions:
2 Fields:
Translation:
AnimalsCells
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effect of OATP1B transporter inhibition on the pharmacokinetics of atorvastatin in healthy volunteers. Clin Pharmacol Ther. 2007 Feb; 81(2):194-204.
Lau YY, Huang Y, Frassetto L, Benet LZ. PMID: 17192770.
View in:
PubMed Mentions:
106 Fields:
Translation:
HumansCells
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Elucidating the effect of final-day dosing of rifampin in induction studies on hepatic drug disposition and metabolism. J Pharmacol Exp Ther. 2006 Nov; 319(2):864-70.
Lam JL, Shugarts SB, Okochi H, Benet LZ. PMID: 16905688.
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PubMed Mentions:
11 Fields:
Translation:
AnimalsCells
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In vitro and in vivo correlation of hepatic transporter effects on erythromycin metabolism: characterizing the importance of transporter-enzyme interplay. Drug Metab Dispos. 2006 Aug; 34(8):1336-44.
Lam JL, Okochi H, Huang Y, Benet LZ. PMID: 16698890.
View in:
PubMed Mentions:
18 Fields:
Translation:
AnimalsCells
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Pharmacokinetics of atorvastatin and its hydroxy metabolites in rats and the effects of concomitant rifampicin single doses: relevance of first-pass effect from hepatic uptake transporters, and intestinal and hepatic metabolism. Drug Metab Dispos. 2006 Jul; 34(7):1175-81.
Lau YY, Okochi H, Huang Y, Benet LZ. PMID: 16624870.
View in:
PubMed Mentions:
36 Fields:
Translation:
AnimalsCells
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Quinacrine is mainly metabolized to mono-desethyl quinacrine by CYP3A4/5 and its brain accumulation is limited by P-glycoprotein. Drug Metab Dispos. 2006 Jul; 34(7):1136-44.
Huang Y, Okochi H, May BC, Legname G, Prusiner SB, Benet LZ, Guglielmo BJ, Lin ET. PMID: 16581945.
View in:
PubMed Mentions:
16 Fields:
Translation:
HumansAnimalsCells
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Liquid chromatographic tandem mass spectrometric assay for the uremic toxin 3-carboxy-4-methyl-5-propyl-2-furanpropionic acid in human plasma. Rapid Commun Mass Spectrom. 2006; 20(10):1611-4.
Huang Y, Sun H, Frassetto L, Benet LZ, Lin ET. PMID: 16628600.
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PubMed Mentions:
2 Fields:
Translation:
Humans
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A cysteine protease inhibitor protects dogs from cardiac damage during infection by Trypanosoma cruzi. Antimicrob Agents Chemother. 2005 Dec; 49(12):5160-1.
Barr SC, Warner KL, Kornreic BG, Piscitelli J, Wolfe A, Benet L, McKerrow JH. PMID: 16304193; PMCID: PMC1315979.
View in:
PubMed Mentions:
59 Fields:
Translation:
Animals
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In vitro and in vivo studies on acyl-coenzyme A-dependent bioactivation of zomepirac in rats. Chem Res Toxicol. 2005 Nov; 18(11):1729-36.
Olsen J, Li C, Bjørnsdottir I, Sidenius U, Hansen SH, Benet LZ. PMID: 16300382.
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PubMed Mentions:
5 Fields:
Translation:
AnimalsCells
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Multiple transporters affect the disposition of atorvastatin and its two active hydroxy metabolites: application of in vitro and ex situ systems. J Pharmacol Exp Ther. 2006 Feb; 316(2):762-71.
Lau YY, Okochi H, Huang Y, Benet LZ. PMID: 16258024.
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PubMed Mentions:
32 Fields:
Translation:
AnimalsCells
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Glucuronidation and the transport of the glucuronide metabolites in LLC-PK1 cells. Mol Pharm. 2005 Sep-Oct; 2(5):428-34.
Chang JH, Benet LZ. PMID: 16196496.
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PubMed Mentions:
3 Fields:
Translation:
HumansAnimalsCells
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Effects of renal failure on drug transport and metabolism. Pharmacol Ther. 2006 Jan; 109(1-2):1-11.
Sun H, Frassetto L, Benet LZ. PMID: 16085315.
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PubMed Mentions:
93 Fields:
Translation:
HumansAnimals
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Effects of short-term alendronate on bone mineral density in haemodialysis patients. Nephrology (Carlton). 2005 Aug; 10(4):393-9.
Wetmore JB, Benet LZ, Kleinstuck D, Frassetto L. PMID: 16109088.
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PubMed Mentions:
11 Fields:
Translation:
Humans
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Cyclosporine pharmacokinetics and dosing modifications in human immunodeficiency virus-infected liver and kidney transplant recipients. Transplantation. 2005 Jul 15; 80(1):13-7.
Frassetto L, Baluom M, Jacobsen W, Christians U, Roland ME, Stock PG, Carlson L, Benet LZ. PMID: 16003227.
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PubMed Mentions:
18 Fields:
Translation:
Humans
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Effect of the MDR1 C3435T variant and P-glycoprotein induction on dicloxacillin pharmacokinetics. J Clin Pharmacol. 2005 Apr; 45(4):411-21.
Putnam WS, Woo JM, Huang Y, Benet LZ. PMID: 15778422.
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PubMed Mentions:
8 Fields:
Translation:
Humans
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There are no useful CYP3A probes that quantitatively predict the in vivo kinetics of other CYP3A substrates and no expectation that one will be found. Mol Interv. 2005 Apr; 5(2):79-83.
Benet LZ. PMID: 15821156.
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PubMed Mentions:
9 Fields:
Translation:
HumansCells
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Basic pharmacological interactions and how they may impact on one another. J Acquir Immune Defic Syndr. 2005 Mar; 38 Suppl 1:S22-3.
Benet L. PMID: 15867606.
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PubMed Mentions: Fields:
Translation:
Humans
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Predicting drug disposition via application of BCS: transport/absorption/ elimination interplay and development of a biopharmaceutics drug disposition classification system. Pharm Res. 2005 Jan; 22(1):11-23.
Wu CY, Benet LZ. PMID: 15771225.
View in:
PubMed Mentions:
279 Fields:
Translation:
HumansAnimals
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Stereoselective taurine conjugation of (R)-benoxaprofen enantiomer in rats: in vivo and in vitro studies using rat hepatic mitochondria and microsomes. Pharm Res. 2005 Jan; 22(1):79-85.
Mohri K, Okada K, Benet LZ. PMID: 15771233.
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PubMed Mentions: Fields:
Translation:
AnimalsCells
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Hepatic microsome studies are insufficient to characterize in vivo hepatic metabolic clearance and metabolic drug-drug interactions: studies of digoxin metabolism in primary rat hepatocytes versus microsomes. Drug Metab Dispos. 2004 Nov; 32(11):1311-6.
Lam JL, Benet LZ. PMID: 15483198.
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PubMed Mentions:
15 Fields:
Translation:
AnimalsCells
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Automated, fast, and sensitive quantification of drugs in human plasma by LC/LC-MS: quantification of 6 protease inhibitors and 3 nonnucleoside transcriptase inhibitors. Ther Drug Monit. 2004 Oct; 26(5):546-62.
Egge-Jacobsen W, Unger M, Niemann CU, Baluom M, Hirai S, Benet LZ, Christians U. PMID: 15385839.
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PubMed Mentions:
2 Fields:
Translation:
Humans
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Novel percutaneous adventitial drug delivery system for regional vascular treatment. Catheter Cardiovasc Interv. 2004 Oct; 63(2):222-30.
Ikeno F, Lyons J, Kaneda H, Baluom M, Benet LZ, Rezaee M. PMID: 15390346.
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PubMed Mentions:
5 Fields:
Translation:
Animals
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Alterations in glucose metabolism by cyclosporine in rat brain slices link to oxidative stress: interactions with mTOR inhibitors. Br J Pharmacol. 2004 Oct; 143(3):388-96.
Christians U, Gottschalk S, Miljus J, Hainz C, Benet LZ, Leibfritz D, Serkova N. PMID: 15339861; PMCID: PMC1575349.
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PubMed Mentions:
21 Fields:
Translation:
AnimalsCells
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Effects of uremic toxins on hepatic uptake and metabolism of erythromycin. Drug Metab Dispos. 2004 Nov; 32(11):1239-46.
Sun H, Huang Y, Frassetto L, Benet LZ. PMID: 15286055.
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PubMed Mentions:
31 Fields:
Translation:
AnimalsCells
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P-glycoprotein (P-gp/MDR1)-mediated efflux of sex-steroid hormones and modulation of P-gp expression in vitro. Pharm Res. 2004 Jul; 21(7):1284-93.
Kim WY, Benet LZ. PMID: 15290871.
View in:
PubMed Mentions:
36 Fields:
Translation:
HumansAnimalsCells
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Unmasking the dynamic interplay between efflux transporters and metabolic enzymes. Int J Pharm. 2004 Jun 11; 277(1-2):3-9.
Benet LZ, Cummins CL, Wu CY. PMID: 15158963.
View in:
PubMed Mentions:
57 Fields:
Translation:
HumansAnimals
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Pharmacogenomics and transplantation: where are we? Am J Transplant. 2004 Jun; 4(6):843.
Frassetto LA, Benet LZ. PMID: 15147415.
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PubMed Mentions: Fields:
Translation:
Humans
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Biochemical mechanisms of cyclosporine neurotoxicity. Mol Interv. 2004 Apr; 4(2):97-107.
Serkova NJ, Christians U, Benet LZ. PMID: 15087483.
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PubMed Mentions:
37 Fields:
Translation:
HumansAnimals
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Ex situ inhibition of hepatic uptake and efflux significantly changes metabolism: hepatic enzyme-transporter interplay. J Pharmacol Exp Ther. 2004 Mar; 308(3):1040-5.
Lau YY, Wu CY, Okochi H, Benet LZ. PMID: 14634033.
View in:
PubMed Mentions:
18 Fields:
Translation:
Animals
-
Disposition of tacrolimus in isolated perfused rat liver: influence of troleandomycin, cyclosporine, and gg918. Drug Metab Dispos. 2003 Nov; 31(11):1292-5.
Wu CY, Benet LZ. PMID: 14570757.
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PubMed Mentions:
15 Fields:
Translation:
Animals
-
CYP3A4-transfected Caco-2 cells as a tool for understanding biochemical absorption barriers: studies with sirolimus and midazolam. J Pharmacol Exp Ther. 2004 Jan; 308(1):143-55.
Cummins CL, Jacobsen W, Christians U, Benet LZ. PMID: 14569063.
View in:
PubMed Mentions:
22 Fields:
Translation:
HumansAnimalsCells
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Transporter-enzyme interactions: implications for predicting drug-drug interactions from in vitro data. Curr Drug Metab. 2003 Oct; 4(5):393-8.
Benet LZ, Cummins CL, Wu CY. PMID: 14529371.
View in:
PubMed Mentions:
38 Fields:
Translation:
HumansAnimals
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Covalent binding of 2-phenylpropionyl-S-acyl-CoA thioester to tissue proteins in vitro. Drug Metab Dispos. 2003 Jun; 31(6):727-30.
Li C, Olurinde MO, Hodges LM, Grillo MP, Benet LZ. PMID: 12756204.
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PubMed Mentions: Fields:
Translation:
HumansAnimalsCells
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In vivo mechanistic studies on the metabolic activation of 2-phenylpropionic acid in rat. J Pharmacol Exp Ther. 2003 Apr; 305(1):250-6.
Li C, Grillo MP, Benet LZ. PMID: 12649376.
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PubMed Mentions:
2 Fields:
Translation:
Animals
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In vivo modulation of intestinal CYP3A metabolism by P-glycoprotein: studies using the rat single-pass intestinal perfusion model. J Pharmacol Exp Ther. 2003 Apr; 305(1):306-14.
Cummins CL, Salphati L, Reid MJ, Benet LZ. PMID: 12649383.
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PubMed Mentions:
27 Fields:
Translation:
Animals
-
In vitro studies on the chemical reactivity of 2,4-dichlorophenoxyacetyl-S-acyl-CoA thioester. Toxicol Appl Pharmacol. 2003 Mar 01; 187(2):101-9.
Li C, Grillo MP, Benet LZ. PMID: 12649042.
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PubMed Mentions:
4 Fields:
Translation:
HumansAnimalsCells
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Pharmacokinetics of cyclosporine pre- and post-liver transplantation. J Clin Pharmacol. 2003 Jan; 43(1):38-42.
Hebert MF, Wacher VJ, Roberts JP, Benet LZ. PMID: 12520626.
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PubMed Mentions: Fields:
Translation:
HumansCTClinical Trials
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Pharmacokinetic interactions between cyclosporine and protease inhibitors in HIV+ subjects. Drug Metab Pharmacokinet. 2003; 18(2):114-20.
Frassetto L, Thai T, Aggarwal AM, Bucher P, Jacobsen W, Christians U, Benet LZ, Floren LC. PMID: 15618725.
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PubMed Mentions:
6 Fields:
-
Inhibition of cytochrome P450 3A4 by extracts and kavalactones of Piper methysticum (Kava-Kava). Planta Med. 2002 Dec; 68(12):1055-8.
Unger M, Holzgrabe U, Jacobsen W, Cummins C, Benet LZ. PMID: 12494328.
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PubMed Mentions:
12 Fields:
Translation:
AnimalsCells
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Functional characterization of monocarboxylic acid, large neutral amino acid, bile acid and peptide transporters, and P-glycoprotein in MDCK and Caco-2 cells. J Pharm Sci. 2002 Dec; 91(12):2622-35.
Putnam WS, Ramanathan S, Pan L, Takahashi LH, Benet LZ. PMID: 12434407.
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PubMed Mentions:
14 Fields:
Translation:
HumansAnimalsCells
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Enantioselective covalent binding of 2-phenylpropionic Acid to protein in vitro in rat hepatocytes. Chem Res Toxicol. 2002 Nov; 15(11):1480-7.
Li C, Benet LZ, Grillo MP. PMID: 12437340.
View in:
PubMed Mentions:
2 Fields:
Translation:
AnimalsCells
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Sex-related differences in the clearance of cytochrome P450 3A4 substrates may be caused by P-glycoprotein. Clin Pharmacol Ther. 2002 Nov; 72(5):474-89.
Cummins CL, Wu CY, Benet LZ. PMID: 12426511.
View in:
PubMed Mentions:
32 Fields:
Translation:
HumansAnimals
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Studies on the chemical reactivity of 2-phenylpropionic acid 1-O-acyl glucuronide and S-acyl-CoA thioester metabolites. Chem Res Toxicol. 2002 Oct; 15(10):1309-17.
Li C, Benet LZ, Grillo MP. PMID: 12387630.
View in:
PubMed Mentions:
7 Fields:
Translation:
Animals
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Close association between the reduction in myocardial energy metabolism and infarct size: dose-response assessment of cyclosporine. J Pharmacol Exp Ther. 2002 Sep; 302(3):1123-8.
Niemann CU, Saeed M, Akbari H, Jacobsen W, Benet LZ, Christians U, Serkova N. PMID: 12183671.
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PubMed Mentions:
11 Fields:
Translation:
AnimalsCells
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Contributions of saturable active secretion, passive transcellular, and paracellular diffusion to the overall transport of furosemide across adenocarcinoma (Caco-2) cells. J Pharm Sci. 2002 Apr; 91(4):1169-77.
Flanagan SD, Takahashi LH, Liu X, Benet LZ. PMID: 11948555.
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PubMed Mentions:
12 Fields:
Translation:
HumansCells
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Can the enhanced renal clearance of antibiotics in cystic fibrosis patients be explained by P-glycoprotein transport? Pharm Res. 2002 Apr; 19(4):457-62.
Susanto M, Benet LZ. PMID: 12033380.
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PubMed Mentions:
19 Fields:
Translation:
HumansCells
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Effect of calcineurin inhibitor therapy on P-gp expression and function in lymphocytes of renal transplant patients: a preliminary evaluation. J Clin Pharmacol. 2002 Mar; 42(3):304-11.
Parasrampuria DA, Lantz MV, Birnbaum JL, Vincenti FG, Benet LZ. PMID: 11865967.
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PubMed Mentions:
2 Fields:
Translation:
HumansCells
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Comparison of the effects of cyclosporin a on the metabolism of perfused rat brain slices during normoxia and hypoxia. J Cereb Blood Flow Metab. 2002 Mar; 22(3):342-52.
Serkova N, Donohoe P, Gottschalk S, Hainz C, Niemann CU, Bickler PE, Litt L, Benet LZ, Leibfritz D, Christians U. PMID: 11891440.
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PubMed Mentions:
6 Fields:
Translation:
AnimalsCells
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Changes in plasma protein binding have little clinical relevance. Clin Pharmacol Ther. 2002 Mar; 71(3):115-21.
Benet LZ, Hoener BA. PMID: 11907485.
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PubMed Mentions:
185 Fields:
Translation:
Humans
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Unmasking the dynamic interplay between intestinal P-glycoprotein and CYP3A4. J Pharmacol Exp Ther. 2002 Mar; 300(3):1036-45.
Cummins CL, Jacobsen W, Benet LZ. PMID: 11861813.
View in:
PubMed Mentions:
50 Fields:
Translation:
HumansCells
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Quantitative liquid chromatography-mass spectrometry determination of isatin in urine using automated on-line extraction. J Chromatogr B Analyt Technol Biomed Life Sci. 2002 Feb 15; 767(2):245-53.
Unger M, Jacobsen W, Holzgrabe U, Benet LZ. PMID: 11885853.
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PubMed Mentions:
1 Fields:
Translation:
Humans
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Mechanisms of clinically relevant drug interactions associated with tacrolimus. Clin Pharmacokinet. 2002; 41(11):813-51.
Christians U, Jacobsen W, Benet LZ, Lampen A. PMID: 12190331.
View in:
PubMed Mentions:
93 Fields:
Translation:
Humans
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Studies on the reactivity of clofibryl-S-acyl-CoA thioester with glutathione in vitro. Drug Metab Dispos. 2002 Jan; 30(1):55-62.
Grillo MP, Benet LZ. PMID: 11744612.
View in:
PubMed Mentions:
5 Fields:
Translation:
AnimalsCells
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Comparison of furosemide and vinblastine secretion from cell lines overexpressing multidrug resistance protein (P-glycoprotein) and multidrug resistance-associated proteins (MRP1 and MRP2). Pharmacology. 2002; 64(3):126-34.
Flanagan SD, Cummins CL, Susanto M, Liu X, Takahashi LH, Benet LZ. PMID: 11834888.
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PubMed Mentions:
12 Fields:
Translation:
AnimalsCells
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Comparison of bidirectional cephalexin transport across MDCK and caco-2 cell monolayers: interactions with peptide transporters. Pharm Res. 2002 Jan; 19(1):27-33.
Putnam WS, Pan L, Tsutsui K, Takahashi L, Benet LZ. PMID: 11837697.
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PubMed Mentions:
6 Fields:
Translation:
HumansAnimalsCells
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Red wine decreases cyclosporine bioavailability. Clin Pharmacol Ther. 2001 Nov; 70(5):462-7.
Tsunoda SM, Harris RZ, Christians U, Velez RL, Freeman RB, Benet LZ, Warshaw A. PMID: 11719733.
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PubMed Mentions:
7 Fields:
Translation:
HumansCTClinical Trials
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The drug efflux-metabolism alliance: biochemical aspects. Adv Drug Deliv Rev. 2001 Oct 01; 50 Suppl 1:S3-11.
Benet LZ, Cummins CL. PMID: 11576692.
View in:
PubMed Mentions:
34 Fields:
Translation:
HumansAnimals
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Effect of alpha-fluorination of valproic acid on valproyl-S-acyl-CoA formation in vivo in rats. Drug Metab Dispos. 2001 Sep; 29(9):1210-5.
Grillo MP, Chiellini G, Tonelli M, Benet LZ. PMID: 11502730.
View in:
PubMed Mentions:
5 Fields:
Translation:
Animals
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Interaction of gamma-glutamyltranspeptidase with clofibryl-S-acyl-glutathione in vitro and in vivo in rat. Chem Res Toxicol. 2001 Aug; 14(8):1033-40.
Grillo MP, Benet LZ. PMID: 11511177.
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PubMed Mentions: Fields:
Translation:
AnimalsCells
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Characterizing the expression of CYP3A4 and efflux transporters (P-gp, MRP1, and MRP2) in CYP3A4-transfected Caco-2 cells after induction with sodium butyrate and the phorbol ester 12-O-tetradecanoylphorbol-13-acetate. Pharm Res. 2001 Aug; 18(8):1102-9.
Cummins CL, Mangravite LM, Benet LZ. PMID: 11587480.
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PubMed Mentions:
19 Fields:
Translation:
HumansCells
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Sirolimus, but not the structurally related RAD (everolimus), enhances the negative effects of cyclosporine on mitochondrial metabolism in the rat brain. Br J Pharmacol. 2001 Jul; 133(6):875-85.
Serkova N, Jacobsen W, Niemann CU, Litt L, Benet LZ, Leibfritz D, Christians U. PMID: 11454661; PMCID: PMC1572850.
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PubMed Mentions:
24 Fields:
Translation:
AnimalsCells
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Metabolism of sirolimus and its derivative everolimus by cytochrome P450 3A4: insights from docking, molecular dynamics, and quantum chemical calculations. J Med Chem. 2001 Jun 07; 44(12):2027-34.
Kuhn B, Jacobsen W, Christians U, Benet LZ, Kollman PA. PMID: 11384247.
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PubMed Mentions:
8 Fields:
Translation:
Cells
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Active secretion and enterocytic drug metabolism barriers to drug absorption. Adv Drug Deliv Rev. 2001 Mar 01; 46(1-3):89-102.
Wacher VJ, Salphati L, Benet LZ. PMID: 11259835.
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PubMed Mentions:
60 Fields:
Translation:
HumansAnimalsCells
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Membrane transport of mycophenolate mofetil and its active metabolite, mycophenolic acid in MDCK and MDR1-MDCK cell monolayers. J Heart Lung Transplant. 2001 Feb; 20(2):234-235.
Sawamoto T, Van Gelder T, Christians U, Okamura N, Jacobsen W, Benet L. PMID: 11250452.
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PubMed Mentions:
6 Fields:
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Comparison of the in vitro metabolism of the macrolide immunosuppressants sirolimus and RAD. Transplant Proc. 2001 Feb-Mar; 33(1-2):514-5.
Jacobsen W, Serkova N, Hausen B, Morris RE, Benet LZ, Christians U. PMID: 11266932.
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PubMed Mentions:
30 Fields:
Translation:
HumansCells
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The gut as a barrier to drug absorption: combined role of cytochrome P450 3A and P-glycoprotein. Clin Pharmacokinet. 2001; 40(3):159-68.
Zhang Y, Benet LZ. PMID: 11327196.
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PubMed Mentions:
91 Fields:
Translation:
HumansAnimals
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The pharmacokinetics and metabolic disposition of tacrolimus: a comparison across ethnic groups. Clin Pharmacol Ther. 2001 Jan; 69(1):24-31.
Mancinelli LM, Frassetto L, Floren LC, Dressler D, Carrier S, Bekersky I, Benet LZ, Christians U. PMID: 11180035.
View in:
PubMed Mentions:
56 Fields:
Translation:
HumansCTClinical Trials
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Identification of hepatic protein targets of the reactive metabolites of the non-hepatotoxic regioisomer of acetaminophen, 3'-hydroxyacetanilide, in the mouse in vivo using two-dimensional gel electrophoresis and mass spectrometry. Adv Exp Med Biol. 2001; 500:663-73.
Qiu Y, Benet LZ, Burlingame AL. PMID: 11765013.
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PubMed Mentions:
27 Fields:
Translation:
Animals
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A human lymphocyte based ex vivo assay to study the effect of drugs on P-glycoprotein (P-gp) function. Pharm Res. 2001 Jan; 18(1):39-44.
Parasrampuria DA, Lantz MV, Benet LZ. PMID: 11336351.
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PubMed Mentions:
6 Fields:
Translation:
HumansCells
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Chiral bioequivalence: effect of absorption rate on racemic etodolac. Clin Pharmacokinet. 2000 Dec; 39(6):459-69.
Boni JR, Korth-Bradley JM, Richards LS, Chiang ST, Hicks DR, Benet LZ. PMID: 11192477.
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PubMed Mentions:
3 Fields:
Translation:
HumansCTClinical Trials
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Lactonization is the critical first step in the disposition of the 3-hydroxy-3-methylglutaryl-CoA reductase inhibitor atorvastatin. Drug Metab Dispos. 2000 Nov; 28(11):1369-78.
Jacobsen W, Kuhn B, Soldner A, Kirchner G, Sewing KF, Kollman PA, Benet LZ, Christians U. PMID: 11038166.
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PubMed Mentions:
69 Fields:
Translation:
HumansCells
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In vitro evaluation of the disposition of A novel cysteine protease inhibitor. Drug Metab Dispos. 2000 Nov; 28(11):1343-51.
Jacobsen W, Christians U, Benet LZ. PMID: 11038163.
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PubMed Mentions:
24 Fields:
Translation:
HumansCells
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Automated, fast and sensitive quantification of drugs in blood by liquid chromatography-mass spectrometry with on-line extraction: immunosuppressants. J Chromatogr B Biomed Sci Appl. 2000 Oct 01; 748(1):41-53.
Christians U, Jacobsen W, Serkova N, Benet LZ, Vidal C, Sewing KF, Manns MP, Kirchner GI. PMID: 11092585.
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PubMed Mentions:
25 Fields:
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Tissue distribution and clinical monitoring of the novel macrolide immunosuppressant SDZ-RAD and its metabolites in monkey lung transplant recipients: interaction with cyclosporine. J Pharmacol Exp Ther. 2000 Jul; 294(1):323-32.
Serkova N, Hausen B, Berry GJ, Jacobsen W, Benet LZ, Morris RE, Christians U. PMID: 10871329.
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PubMed Mentions:
11 Fields:
Translation:
Animals
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Recommendations for bioequivalence testing of cyclosporine generics revisited. Ther Drug Monit. 2000 Jun; 22(3):330-45.
Christians U, First MR, Benet LZ. PMID: 10850403.
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PubMed Mentions:
8 Fields:
Translation:
Humans
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Active transport of the angiotensin-II antagonist losartan and its main metabolite EXP 3174 across MDCK-MDR1 and caco-2 cell monolayers. Br J Pharmacol. 2000 Mar; 129(6):1235-43.
Soldner A, Benet LZ, Mutschler E, Christians U. PMID: 10725273; PMCID: PMC1571937.
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PubMed Mentions:
26 Fields:
Translation:
HumansAnimalsCells
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The novel immunosuppressant SDZ-RAD protects rat brain slices from cyclosporine-induced reduction of high-energy phosphates. Br J Pharmacol. 2000 Feb; 129(3):485-92.
Serkova N, Litt L, Leibfritz D, Hausen B, Morris RE, James TL, Benet LZ, Christians U. PMID: 10711346; PMCID: PMC1571863.
View in:
PubMed Mentions:
8 Fields:
Translation:
AnimalsCells
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Combined immunosuppression with cyclosporine (neoral) and SDZ RAD in non-human primate lung transplantation: systematic pharmacokinetic-based trials to improve efficacy and tolerability. Transplantation. 2000 Jan 15; 69(1):76-86.
Hausen B, Ikonen T, Briffa N, Berry GJ, Christians U, Robbins RC, Hook L, Serkova N, Benet LZ, Schuler W, Morris RE. PMID: 10653384.
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PubMed Mentions:
6 Fields:
Translation:
Animals
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Ethynylestradiol-mediated induction of hepatic CYP3A9 in female rats: implication for cyclosporine metabolism. Drug Metab Dispos. 1999 Dec; 27(12):1505-11.
Jäger W, Correia MA, Bornheim LM, Mahnke A, Hanstein WG, Xue L, Benet LZ. PMID: 10570034.
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PubMed Mentions:
5 Fields:
Translation:
AnimalsCells
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Intestinal MDR transport proteins and P-450 enzymes as barriers to oral drug delivery. J Control Release. 1999 Nov 01; 62(1-2):25-31.
Benet LZ, Izumi T, Zhang Y, Silverman JA, Wacher VJ. PMID: 10518631.
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PubMed Mentions:
53 Fields:
Translation:
AnimalsCells
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Small intestinal metabolism of the 3-hydroxy-3-methylglutaryl-coenzyme A reductase inhibitor lovastatin and comparison with pravastatin. J Pharmacol Exp Ther. 1999 Oct; 291(1):131-9.
Jacobsen W, Kirchner G, Hallensleben K, Mancinelli L, Deters M, Hackbarth I, Baner K, Benet LZ, Sewing KF, Christians U. PMID: 10490896.
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PubMed Mentions:
11 Fields:
Translation:
HumansAnimalsCells
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Photoinduced covalent binding of frusemide and frusemide glucuronide to human serum albumin. Br J Clin Pharmacol. 1999 Jul; 48(1):79-87.
Mizuma T, McDonagh AF, Lin ET, Benet LZ. PMID: 10383564; PMCID: PMC2014883.
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PubMed Mentions:
1 Fields:
Translation:
HumansCells
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Understanding bioequivalence testing. Transplant Proc. 1999 May; 31(3A Suppl):7S-9S.
Benet LZ. PMID: 10330950.
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PubMed Mentions:
2 Fields:
Translation:
Humans
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Evaluation of individual and combined neurotoxicity of the immunosuppressants cyclosporine and sirolimus by in vitro multinuclear NMR spectroscopy. J Pharmacol Exp Ther. 1999 May; 289(2):800-6.
Serkova N, Litt L, James TL, Sadée W, Leibfritz D, Benet LZ, Christians U. PMID: 10215655.
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PubMed Mentions:
8 Fields:
Translation:
HumansAnimalsCells
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Relevance of pharmacokinetics in narrow therapeutic index drugs. Transplant Proc. 1999 May; 31(3):1642-4; discussion 1675-84.
Benet LZ. PMID: 10331032.
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PubMed Mentions:
5 Fields:
Translation:
Humans
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Coadministration of neoral and the novel rapamycin analog, SDZ RAD, to rat lung allograft recipients: potentiation of immunosuppressive efficacy and improvement of tolerability of staggered versus simultaneous treatment. Transplantation. 1999 Apr 15; 67(7):956-62.
Hausen B, Boeke K, Berry GJ, Segarra I, Benet LZ, Christians U, Morris RE. PMID: 10221478.
View in:
PubMed Mentions:
2 Fields:
Translation:
Animals
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Grapefruit juice activates P-glycoprotein-mediated drug transport. Pharm Res. 1999 Apr; 16(4):478-85.
Soldner A, Christians U, Susanto M, Wacher VJ, Silverman JA, Benet LZ. PMID: 10227700.
View in:
PubMed Mentions:
31 Fields:
Translation:
HumansAnimalsCells
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Interaction of human serum albumin with furosemide glucuronide: a role of albumin in isomerization, hydrolysis, reversible binding and irreversible binding of a 1-O-acyl glucuronide metabolite. Biopharm Drug Dispos. 1999 Apr; 20(3):131-6.
Mizuma T, Benet LZ, Lin ET. PMID: 10211865.
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PubMed Mentions:
2 Fields:
Translation:
HumansCells
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In vitro biotransformation of a novel antimalarial cysteine protease inhibitor in human liver microsomes. Pharmacology. 1999 Mar; 58(3):147-59.
Zhang Y, Guo X, Lin ET, Benet LZ. PMID: 9925971.
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PubMed Mentions:
2 Fields:
Translation:
HumansAnimalsCells
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Molecular and physical mechanisms of first-pass extraction. Drug Metab Dispos. 1999 Feb; 27(2):161-6.
Hall SD, Thummel KE, Watkins PB, Lown KS, Benet LZ, Paine MF, Mayo RR, Turgeon DK, Bailey DG, Fontana RJ, Wrighton SA. PMID: 9929497.
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PubMed Mentions:
48 Fields:
Translation:
HumansAnimals
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Comparison of cytochrome P-450-dependent metabolism and drug interactions of the 3-hydroxy-3-methylglutaryl-CoA reductase inhibitors lovastatin and pravastatin in the liver. Drug Metab Dispos. 1999 Feb; 27(2):173-9.
Jacobsen W, Kirchner G, Hallensleben K, Mancinelli L, Deters M, Hackbarth I, Benet LZ, Sewing KF, Christians U. PMID: 9929499.
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PubMed Mentions:
32 Fields:
Translation:
HumansCells
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Net secretion of furosemide is subject to indomethacin inhibition, as observed in Caco-2 monolayers and excised rat jejunum. Pharm Res. 1999 Feb; 16(2):221-24.
Flanagan SD, Benet LZ. PMID: 10100306.
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PubMed Mentions:
3 Fields:
Translation:
HumansAnimalsCells
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Metabolism of digoxin and digoxigenin digitoxosides in rat liver microsomes: involvement of cytochrome P4503A. Xenobiotica. 1999 Feb; 29(2):171-85.
Salphati L, Benet LZ. PMID: 10199593.
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PubMed Mentions:
12 Fields:
Translation:
HumansAnimalsCells
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Development of a high-performance liquid chromatographic-electrospray mass spectrometric assay for the specific and sensitive quantification of the novel immunosuppressive macrolide 40-O-(2-hydroxyethyl)rapamycin. J Chromatogr B Biomed Sci Appl. 1998 Dec 11; 720(1-2):179-87.
Segarra I, Brazelton TR, Guterman N, Hausen B, Jacobsen W, Morris RE, Benet LZ, Christians U. PMID: 9892080.
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PubMed Mentions:
1 Fields:
Translation:
Humans
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Preliminary evaluation of progestins as inducers of cytochrome P450 3A4 activity in postmenopausal women. J Clin Pharmacol. 1998 Dec; 38(12):1137-43.
Tsunoda SM, Harris RZ, Mroczkowski PJ, Benet LZ. PMID: 11301566.
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PubMed Mentions:
4 Fields:
Translation:
HumansCTClinical Trials
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Role of P-glycoprotein and cytochrome P450 3A in limiting oral absorption of peptides and peptidomimetics. J Pharm Sci. 1998 Nov; 87(11):1322-30.
Wacher VJ, Silverman JA, Zhang Y, Benet LZ. PMID: 9811484.
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PubMed Mentions:
82 Fields:
Translation:
Humans
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High-performance liquid chromatographic determination and identification of acyl migration and photodegradation products of furosemide 1-O-acyl glucuronide. J Chromatogr B Biomed Sci Appl. 1998 Oct 23; 718(1):153-62.
Mizuma T, Benet LZ, Lin ET. PMID: 9832372.
View in:
PubMed Mentions:
1 Fields:
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Effects of ketoconazole on the intestinal metabolism, transport and oral bioavailability of K02, a novel vinylsulfone peptidomimetic cysteine protease inhibitor and a P450 3A, P-glycoprotein dual substrate, in male Sprague-Dawley rats. J Pharmacol Exp Ther. 1998 Oct; 287(1):246-52.
Zhang Y, Hsieh Y, Izumi T, Lin ET, Benet LZ. PMID: 9765344.
View in:
PubMed Mentions:
11 Fields:
Translation:
AnimalsCells
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Characterization of P-glycoprotein mediated transport of K02, a novel vinylsulfone peptidomimetic cysteine protease inhibitor, across MDR1-MDCK and Caco-2 cell monolayers. Pharm Res. 1998 Oct; 15(10):1520-4.
Zhang Y, Benet LZ. PMID: 9794492.
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PubMed Mentions:
7 Fields:
Translation:
HumansAnimalsCells
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Impact of intraindividual variability of drugs on therapeutic outcomes: lessons from outside transplantation. Transplant Proc. 1998 Aug; 30(5):1650-1.
Benet LZ. PMID: 9723227.
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PubMed Mentions:
2 Fields:
Translation:
Humans
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Identification of the hepatic protein targets of reactive metabolites of acetaminophen in vivo in mice using two-dimensional gel electrophoresis and mass spectrometry. J Biol Chem. 1998 Jul 10; 273(28):17940-53.
Qiu Y, Benet LZ, Burlingame AL. PMID: 9651401.
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PubMed Mentions:
98 Fields:
Translation:
AnimalsCells
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Metabolism and transport of the macrolide immunosuppressant sirolimus in the small intestine. J Pharmacol Exp Ther. 1998 Jun; 285(3):1104-12.
Lampen A, Zhang Y, Hackbarth I, Benet LZ, Sewing KF, Christians U. PMID: 9618413.
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PubMed Mentions:
32 Fields:
Translation:
HumansAnimalsCells
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Effects of ketoconazole on digoxin absorption and disposition in rat. Pharmacology. 1998 Jun; 56(6):308-13.
Salphati L, Benet LZ. PMID: 9654217.
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PubMed Mentions:
6 Fields:
Translation:
Animals
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Stereoselective metabolism of benoxaprofen in rats. Biliary excretion of benoxaprofen taurine conjugate and glucuronide. Drug Metab Dispos. 1998 Apr; 26(4):332-7.
Mohri K, Okada K, Benet LZ. PMID: 9531520.
View in:
PubMed Mentions:
4 Fields:
Translation:
Animals
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Overlapping substrate specificities of cytochrome P450 3A and P-glycoprotein for a novel cysteine protease inhibitor. Drug Metab Dispos. 1998 Apr; 26(4):360-6.
Zhang Y, Guo X, Lin ET, Benet LZ. PMID: 9531525.
View in:
PubMed Mentions:
15 Fields:
Translation:
HumansAnimalsCells
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Antiprogestin-mediated inactivation of cytochrome P450 3A4. Pharmacology. 1998 Mar; 56(3):150-7.
Jang GR, Benet LZ. PMID: 9532615.
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PubMed Mentions:
4 Fields:
Translation:
HumansCells
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Mechanisms for covalent binding of benoxaprofen glucuronide to human serum albumin. Studies By tandem mass spectrometry. Drug Metab Dispos. 1998 Mar; 26(3):246-56.
Qiu Y, Burlingame AL, Benet LZ. PMID: 9492388.
View in:
PubMed Mentions:
12 Fields:
Translation:
HumansCells
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Modulation of P-glycoprotein expression by cytochrome P450 3A inducers in male and female rat livers. Biochem Pharmacol. 1998 Feb 15; 55(4):387-95.
Salphati L, Benet LZ. PMID: 9514072.
View in:
PubMed Mentions:
16 Fields:
Translation:
Animals
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Preparative chromatography of furosemide 1-O-acyl-glucuronide from urine using micronized amberiite XAD-2 and its application to other 1-O-acyl-glucuronides. Prep Biochem Biotechnol. 1998 Feb; 28(1):37-47.
Mizuma T, Benet LZ, Lin ET. PMID: 9516641.
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PubMed Mentions:
2 Fields:
Translation:
Cells
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Antiprogestin pharmacodynamics, pharmacokinetics, and metabolism: implications for their long-term use. J Pharmacokinet Biopharm. 1997 Dec; 25(6):647-72.
Jang GR, Benet LZ. PMID: 9697076.
View in:
PubMed Mentions:
4 Fields:
Translation:
Humans
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Cytochrome P4503A4-mediated N-demethylation of the antiprogestins lilopristone and onapristone. Drug Metab Dispos. 1997 Oct; 25(10):1119-22.
Jang GR, Benet LZ. PMID: 9321513.
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PubMed Mentions:
2 Fields:
Translation:
HumansCells
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Role of intestinal P-glycoprotein (mdr1) in interpatient variation in the oral bioavailability of cyclosporine. Clin Pharmacol Ther. 1997 Sep; 62(3):248-60.
Lown KS, Mayo RR, Leichtman AB, Hsiao HL, Turgeon DK, Schmiedlin-Ren P, Brown MB, Guo W, Rossi SJ, Benet LZ, Watkins PB. PMID: 9333100.
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PubMed Mentions:
134 Fields:
Translation:
Humans
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Tacrolimus oral bioavailability doubles with coadministration of ketoconazole. Clin Pharmacol Ther. 1997 Jul; 62(1):41-9.
Floren LC, Bekersky I, Benet LZ, Mekki Q, Dressler D, Lee JW, Roberts JP, Hebert MF. PMID: 9246018.
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PubMed Mentions:
64 Fields:
Translation:
Humans
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Investigation of aortic CYP3A bioactivation of nitroglycerin in vivo. J Pharmacol Exp Ther. 1997 Jun; 281(3):1499-505.
Yuan R, Sumi M, Benet LZ. PMID: 9190888.
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PubMed Mentions:
7 Fields:
Translation:
Animals
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Stereoselective high-performance liquid chromatography determination of propranolol and 4-hydroxypropranolol in human plasma after pre-column derivatization. J Chromatogr B Biomed Sci Appl. 1997 Apr 25; 692(1):133-40.
Wu ST, Chang YP, Gee WL, Benet LZ, Lin ET. PMID: 9187392.
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PubMed Mentions:
1 Fields:
Translation:
Humans
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Determination of amiprilose in human plasma by high-performance liquid chromatography with fluorimetric detection. J Chromatogr B Biomed Sci Appl. 1997 Apr 25; 692(1):149-56.
Wu ST, Benet LZ, Lin ET. PMID: 9187394.
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PubMed Mentions: Fields:
Translation:
Humans
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Evaluation of orally administered highly variable drugs and drug formulations. Pharm Res. 1996 Nov; 13(11):1590-4.
Shah VP, Yacobi A, Barr WH, Benet LZ, Breimer D, Dobrinska MR, Endrenyi L, Fairweather W, Gillespie W, Gonzalez MA, Hooper J, Jackson A, Lesko LJ, Midha KK, Noonan PK, Patnaik R, Williams RL. PMID: 8956322.
View in:
PubMed Mentions:
22 Fields:
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Pharmacokinetics and pharmacodynamics of metformin in healthy subjects and patients with noninsulin-dependent diabetes mellitus. J Clin Pharmacol. 1996 Nov; 36(11):1012-21.
Sambol NC, Chiang J, O'Conner M, Liu CY, Lin ET, Goodman AM, Benet LZ, Karam JH. PMID: 8973990.
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PubMed Mentions:
50 Fields:
Translation:
HumansCTClinical Trials
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Food intake and dosage level, but not tablet vs solution dosage form, affect the absorption of metformin HCl in man. Br J Clin Pharmacol. 1996 Oct; 42(4):510-2.
Sambol NC, Brookes LG, Chiang J, Goodman AM, Lin ET, Liu CY, Benet LZ. PMID: 8904626.
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PubMed Mentions:
24 Fields:
Translation:
HumansCTClinical Trials
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Morality play. Science. 1996 Sep 27; 273(5283):1782; author reply 1784-5.
Benet LZ. PMID: 8815536.
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PubMed Mentions: Fields:
Translation:
Humans
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Identification of CYP3A4 as the principal enzyme catalyzing mifepristone (RU 486) oxidation in human liver microsomes. Biochem Pharmacol. 1996 Sep 13; 52(5):753-61.
Jang GR, Wrighton SA, Benet LZ. PMID: 8765473.
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PubMed Mentions:
15 Fields:
Translation:
HumansCells
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In vivo depletion of free thiols does not account for nitroglycerin-induced tolerance: a thiol-nitrate interaction hypothesis as an alternative explanation for nitroglycerin activity and tolerance. J Pharmacol Exp Ther. 1996 Sep; 278(3):1296-305.
Haj-Yehia AI, Benet LZ. PMID: 8819515.
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PubMed Mentions:
4 Fields:
Translation:
Animals
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Acute dose-dependent disposition studies of nicotinic acid in rats. Drug Metab Dispos. 1996 Jul; 24(7):773-9.
Iwaki M, Ogiso T, Hayashi H, Tanino T, Benet LZ. PMID: 8818575.
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PubMed Mentions:
4 Fields:
Translation:
AnimalsCells
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Tolerance to nitroglycerin in rabbit aorta. Investigating the involvement of the mu isozyme of glutathione S-transferases. Biochem Pharmacol. 1996 May 17; 51(10):1357-63.
Kenkare SR, Benet LZ. PMID: 8787552.
View in:
PubMed Mentions:
1 Fields:
Translation:
Animals
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Suppression of intestinal and hepatic cytochrome P4503A in murine Toxoplasma infection. Effects of N-acetylcysteine and N(G)-monomethyl-L-arginine on the hepatic suppression. Xenobiotica. 1996 Apr; 26(4):381-94.
Berg-Candolfi M, Candolfi E, Benet LZ. PMID: 9173679.
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PubMed Mentions:
4 Fields:
Translation:
AnimalsCells
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The effects of menopause and hormone replacement therapies on prednisolone and erythromycin pharmacokinetics. Clin Pharmacol Ther. 1996 Apr; 59(4):429-35.
Harris RZ, Tsunoda SM, Mroczkowski P, Wong H, Benet LZ. PMID: 8612388.
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PubMed Mentions:
17 Fields:
Translation:
Humans
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Inhibition of cyclosporine and tetrahydrocannabinol metabolism by cannabidiol in mouse and human microsomes. Xenobiotica. 1996 Mar; 26(3):275-84.
Jaeger W, Benet LZ, Bornheim LM. PMID: 8730919.
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PubMed Mentions:
13 Fields:
Translation:
HumansAnimalsCells
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The effect of water-soluble vitamin E on cyclosporine pharmacokinetics in healthy volunteers. Clin Pharmacol Ther. 1996 Mar; 59(3):297-303.
Chang T, Benet LZ, Hebert MF. PMID: 8653992.
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PubMed Mentions:
20 Fields:
Translation:
HumansCTClinical Trials
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Kidney function and age are both predictors of pharmacokinetics of metformin. J Clin Pharmacol. 1995 Nov; 35(11):1094-102.
Sambol NC, Chiang J, Lin ET, Goodman AM, Liu CY, Benet LZ, Cogan MG. PMID: 8626883.
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PubMed Mentions:
44 Fields:
Translation:
Humans
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Differentiation of absorption and first-pass gut and hepatic metabolism in humans: studies with cyclosporine. Clin Pharmacol Ther. 1995 Nov; 58(5):492-7.
Wu CY, Benet LZ, Hebert MF, Gupta SK, Rowland M, Gomez DY, Wacher VJ. PMID: 7586942.
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PubMed Mentions:
70 Fields:
Translation:
Humans
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Synthesis and mass-spectrometric characterization of human serum albumins modified by covalent binding of two non-steroidal anti-inflammatory drugs: tolmetin and zomepirac. Biochem J. 1995 Oct 15; 311 ( Pt 2):431-5.
Zia-Amirhosseini P, Ding A, Burlingame AL, McDonagh AF, Benet LZ. PMID: 7487878; PMCID: PMC1136018.
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PubMed Mentions:
2 Fields:
Translation:
HumansCells
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Immunopharmacodynamic studies of cyclosporine in patients awaiting renal transplantation. J Clin Pharmacol. 1995 Oct; 35(10):967-73.
d'Uscio CH, Aweeka FT, Prueksaritanont T, Tomlanovich SJ, Gupta SK, Lantz MV, Gambertoglio JG, Garovoy MR, Benet LZ. PMID: 8568014.
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PubMed Mentions:
1 Fields:
Translation:
Humans
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Stereoselective disposition of naproxen glucuronide in the rat. Drug Metab Dispos. 1995 Oct; 23(10):1099-103.
Iwaki M, Bischer A, Nguyen AC, McDonagh AF, Benet LZ. PMID: 8654198.
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PubMed Mentions:
2 Fields:
Translation:
Animals
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Stereoselective reversible binding properties of the glucuronide conjugates of fenoprofen enantiomers to human serum albumin. Drug Metab Dispos. 1995 Sep; 23(9):900-3.
Bischer A, Iwaki M, Zia-Amirhosseini P, Benet LZ. PMID: 8565778.
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PubMed Mentions:
1 Fields:
Translation:
HumansAnimalsCells
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Effect of cannabidiol pretreatment on the kinetics of tetrahydrocannabinol metabolites in mouse brain. Drug Metab Dispos. 1995 Aug; 23(8):825-31.
Bornheim LM, Kim KY, Li J, Perotti BY, Benet LZ. PMID: 7493549.
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PubMed Mentions:
27 Fields:
Translation:
Animals
-
Gender effects in pharmacokinetics and pharmacodynamics. Drugs. 1995 Aug; 50(2):222-39.
Harris RZ, Benet LZ, Schwartz JB. PMID: 8521756.
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PubMed Mentions:
92 Fields:
Translation:
HumansCells
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Stereoselective binding properties of naproxen glucuronide diastereomers to proteins. J Pharmacokinet Biopharm. 1995 Aug; 23(4):379-95.
Bischer A, Zia-Amirhosseini P, Iwaki M, McDonagh AF, Benet LZ. PMID: 8882746.
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PubMed Mentions:
3 Fields:
Translation:
HumansAnimalsCells
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Overlapping substrate specificities and tissue distribution of cytochrome P450 3A and P-glycoprotein: implications for drug delivery and activity in cancer chemotherapy. Mol Carcinog. 1995 Jul; 13(3):129-34.
Wacher VJ, Wu CY, Benet LZ. PMID: 7619215.
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PubMed Mentions:
177 Fields:
Translation:
Humans
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The effects of ketoconazole on the intestinal metabolism and bioavailability of cyclosporine. Clin Pharmacol Ther. 1995 Jul; 58(1):15-9.
Gomez DY, Wacher VJ, Tomlanovich SJ, Hebert MF, Benet LZ. PMID: 7628178.
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PubMed Mentions:
45 Fields:
Translation:
HumansCTClinical Trials
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Bioequivalence and narrow therapeutic index drugs. Pharmacotherapy. 1995 Jul-Aug; 15(4):433-40.
Benet LZ, Goyan JE. PMID: 7479195.
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PubMed Mentions:
10 Fields:
Translation:
Humans
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Time course of cyclosporine and ist motabolites in blood, liver and spleen of naive Lewis rats: comparison with preliminary data obtained in transplanted animals. Biopharm Drug Dispos. 1995 May; 16(4):303-12.
Wacher VJ, Liu T, Roberts JP, Ascher NL, Benet LZ. PMID: 7548779.
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PubMed Mentions: Fields:
Translation:
Animals
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2-(4-N-maleimidophenyl)-6-methoxybenzofuran: a superior derivatizing agent for fluorimetric determination of aliphatic thiols by high-performance liquid chromatography. J Chromatogr B Biomed Appl. 1995 Apr 07; 666(1):45-53.
Haj-Yehia AI, Benet LZ. PMID: 7655620.
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PubMed Mentions: Fields:
Translation:
Animals
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Dissociation of tissue thiols content from nitroglycerin-induced cyclic-3',5'-guanosine monophosphate and the state of tolerance: in vivo experiments in rats. J Pharmacol Exp Ther. 1995 Apr; 273(1):94-100.
Haj-Yehia AI, Benet LZ. PMID: 7714819.
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PubMed Mentions:
2 Fields:
Translation:
Animals
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Biliary excretion of furosemide glucuronide in rabbits. Biol Pharm Bull. 1995 Mar; 18(3):447-53.
Sekikawa H, Yagi N, Oda K, Kenmotsu H, Takada M, Chen HF, Lin ET, Benet LZ. PMID: 7550101.
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PubMed Mentions: Fields:
Translation:
HumansAnimals
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Basic principles of pharmacokinetics. Toxicol Pathol. 1995 Mar-Apr; 23(2):115-23.
Benet LZ, Zia-Amirhosseini P. PMID: 7569664.
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PubMed Mentions:
54 Fields:
Translation:
HumansAnimals
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Reactivity of tolmetin glucuronide with human serum albumin. Identification of binding sites and mechanisms of reaction by tandem mass spectrometry. Drug Metab Dispos. 1995 Mar; 23(3):369-76.
Ding A, Zia-Amirhosseini P, McDonagh AF, Burlingame AL, Benet LZ. PMID: 7628303.
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PubMed Mentions:
11 Fields:
Translation:
HumansCells
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Apparent intramolecular acyl migration and hydrolysis of furosemide glucuronide in aqueous solution. Biol Pharm Bull. 1995 Jan; 18(1):134-9.
Sekikawa H, Yagi N, Lin ET, Benet LZ. PMID: 7735228.
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PubMed Mentions: Fields:
Translation:
HumansCells
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Hypersensitivity to nonsteroidal anti-inflammatory drugs. Nat Med. 1995 Jan; 1(1):2-4.
Zia-Amirhosseini PZ, Harris RZ, Brodsky FM, Benet LZ. PMID: 7584944.
View in:
PubMed Mentions:
4 Fields:
Translation:
Animals
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Determination of aliphatic thiols by fluorometric high-performance liquid chromatography after precolumn derivatization with 2-(4-N-maleimidophenyl)-6-methylbenzothiazole. Pharm Res. 1995 Jan; 12(1):155-60.
Haj-Yehia AI, Benet LZ. PMID: 7724479.
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PubMed Mentions: Fields:
Translation:
Animals
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Correlation of the response to nitroglycerin in rabbit aorta with the activity of the mu class glutathione S-transferase. Biochem Pharmacol. 1994 Dec 16; 48(12):2231-5.
Kenkare SR, Han C, Benet LZ. PMID: 7811305.
View in:
PubMed Mentions:
6 Fields:
Translation:
Animals
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Simultaneous measurement of nicotinic acid and its major metabolite, nicotinuric acid in urine using high-performance liquid chromatography: application of solid-liquid extraction. J Chromatogr B Biomed Appl. 1994 Nov 04; 661(1):154-8.
Iwaki M, Ogiso T, Hayashi H, Lin ET, Benet LZ. PMID: 7866544.
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PubMed Mentions:
1 Fields:
Translation:
Animals
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Irreversible binding of tolmetin to macromolecules via its glucuronide: binding to blood constituents, tissue homogenates and subcellular fractions in vitro. Xenobiotica. 1994 Jun; 24(6):495-506.
Ojingwa JC, Spahn-Langguth H, Benet LZ. PMID: 7975715.
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PubMed Mentions: Fields:
Translation:
HumansAnimalsCells
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HPLC assay for FK 506 and two metabolites in isolated rat hepatocytes and rat liver microsomes. Pharm Res. 1994 Jun; 11(6):844-7.
Perotti BY, Prueksaritanont T, Benet LZ. PMID: 7524055.
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PubMed Mentions:
2 Fields:
Translation:
AnimalsCells
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Menopause: pharmacodynamics and pharmacokinetics. Exp Gerontol. 1994 May-Aug; 29(3-4):437-44.
Gustavson LE, Benet LZ. PMID: 7925762.
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PubMed Mentions:
3 Fields:
Translation:
HumansCTClinical Trials
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Pharmacokinetics of nitroglycerin and its four metabolites during nitroglycerin transdermal administration. Biopharm Drug Dispos. 1994 Mar; 15(2):179-83.
Han C, Jung P, Sanders SW, Lin ET, Benet LZ. PMID: 8011969.
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PubMed Mentions:
4 Fields:
Translation:
HumansCTClinical Trials
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Opportunities for integration of pharmacokinetics, pharmacodynamics, and toxicokinetics in rational drug development. J Clin Pharmacol. 1994 Feb; 34(2):111-9.
Peck CC, Barr WH, Benet LZ, Collins J, Desjardins RE, Furst DE, Harter JG, Levy G, Ludden T, Rodman JH, et al. PMID: 8163710.
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PubMed Mentions:
13 Fields:
Translation:
HumansAnimals
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Reversible binding of tolmetin, zomepirac, and their glucuronide conjugates to human serum albumin and plasma. J Pharmacokinet Biopharm. 1994 Feb; 22(1):19-40.
Ojingwa JC, Spahn-Langguth H, Benet LZ. PMID: 8027947.
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PubMed Mentions:
2 Fields:
Translation:
HumansCells
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Bioactivation by glucuronide-conjugate formation. Adv Pharmacol. 1994; 27:385-97.
Zia-Amirhosseini P, Spahn-Langguth H, Benet LZ. PMID: 8068561.
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PubMed Mentions: Fields:
Translation:
HumansAnimals
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Pharmacokinetics of orally and intravenously administered cyclosporine in pre-kidney transplant patients. J Clin Pharmacol. 1994 Jan; 34(1):60-7.
Aweeka FT, Tomlanovich SJ, Prueksaritanont T, Gupta SK, Benet LZ. PMID: 8132853.
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PubMed Mentions:
7 Fields:
Translation:
Humans
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Pharmacokinetics--a relevant factor for the choice of a drug? Aliment Pharmacol Ther. 1994; 8 Suppl 1:25-32.
Benet LZ, Zech K. PMID: 8180291.
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PubMed Mentions:
14 Fields:
Translation:
HumansCells
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Enhanced covalent binding of tolmetin to proteins in humans after multiple dosing. Clin Pharmacol Ther. 1994 Jan; 55(1):21-7.
Zia-Amirhosseini P, Ojingwa JC, Spahn-Langguth H, McDonagh AF, Benet LZ. PMID: 8299313.
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PubMed Mentions:
2 Fields:
Translation:
HumansCells
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FK 506 metabolism in male and female rat liver microsomes. Drug Metab Dispos. 1994 Jan-Feb; 22(1):85-9.
Perotti BY, Okudaira N, Prueksaritanont T, Benet LZ. PMID: 7512020.
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PubMed Mentions:
4 Fields:
Translation:
AnimalsCells
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Pharmacokinetic profile of etodolac in special populations. Eur J Rheumatol Inflamm. 1994; 14(1):15-8.
Benet LZ. PMID: 7744123.
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PubMed Mentions:
1 Fields:
Translation:
Humans
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Pharmacokinetics and irreversible binding of tolmetin and its glucuronic acid esters in the elderly. Pharmacology. 1993 Nov; 47(5):309-17.
Munafo A, Hyneck ML, Benet LZ. PMID: 8265721.
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Translation:
HumansCells
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Simultaneous pharmacodynamic modeling of the non-steady-state effects of three oral doses of 1,3-glyceryl dinitrate upon blood pressure in healthy volunteers. J Pharmacokinet Biopharm. 1993 Oct; 21(5):515-32.
Gumbleton M, Benet LZ. PMID: 8145129.
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PubMed Mentions:
3 Fields:
Translation:
Humans
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Pharmacokinetics and pharmacodynamics of nitroglycerin and its dinitrate metabolites in conscious dogs: intravenous infusion studies. J Pharmacokinet Biopharm. 1993 Oct; 21(5):533-50.
Lee FW, Salmonson T, Benet LZ. PMID: 8145130.
View in:
PubMed Mentions:
2 Fields:
Translation:
Animals
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Effect of ethacrynic acid, a glutathione-S-transferase inhibitor, on nitroglycerin-mediated cGMP elevation and vasorelaxation of rabbit aortic strips. Biochem Pharmacol. 1993 Jul 20; 46(2):279-84.
Kenkare SR, Benet LZ. PMID: 8394078.
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PubMed Mentions:
3 Fields:
Translation:
Animals
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Cyclosporine metabolism by rat liver microsomes. Evidence for involvement of enzyme(s) other than cytochromes P-450 3A. Drug Metab Dispos. 1993 Jul-Aug; 21(4):730-7.
Prueksaritanont T, Correia MA, Rettie AE, Swinney DC, Thomas PE, Benet LZ. PMID: 8104135.
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PubMed Mentions:
3 Fields:
Translation:
AnimalsCells
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Interpretation and utilization of effect and concentration data collected in an in vivo pharmacokinetic and in vitro pharmacodynamic study. Pharm Res. 1993 Jun; 10(6):889-94.
Gupta SK, Hwang SS, Benet LZ, Gumbleton M. PMID: 8321858.
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PubMed Mentions:
3 Fields:
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Evidence for covalent binding of acyl glucuronides to serum albumin via an imine mechanism as revealed by tandem mass spectrometry. Proc Natl Acad Sci U S A. 1993 May 01; 90(9):3797-801.
Ding A, Ojingwa JC, McDonagh AF, Burlingame AL, Benet LZ. PMID: 8483897; PMCID: PMC46392.
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PubMed Mentions:
15 Fields:
Translation:
HumansCells
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Microsomal acyl glucuronidation: enzyme-kinetic studies with labile glucuronides. Pharmacology. 1993 May; 46(5):268-73.
Spahn-Langguth H, Benet LZ. PMID: 8488171.
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PubMed Mentions:
1 Fields:
Translation:
HumansAnimalsCells
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Nitroglycerin dinitrate metabolites do not affect the pharmacokinetics and pharmacodynamics of nitroglycerin in the dog: a preliminary report. J Pharmacokinet Biopharm. 1993 Apr; 21(2):163-73.
Lee FW, Hu J, Metzler CH, Benet LZ. PMID: 8229678.
View in:
PubMed Mentions:
2 Fields:
Translation:
Animals
-
New techniques in drug metabolism and clinical pharmacology/pharmacokinetics. Am Biotechnol Lab. 1993 Feb; 11(2):44-7.
Benet LZ. PMID: 7763426.
View in:
PubMed Mentions: Fields:
Translation:
HumansAnimals
-
Pharmacokinetics of sustained-release etodolac. Rheumatol Int. 1993; 13(2 Suppl):S3-5.
Benet LZ. PMID: 8210922.
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PubMed Mentions:
1 Fields:
Translation:
Humans
-
In vitro and in vivo irreversible plasma protein binding of beclobric acid enantiomers. Chirality. 1993; 5(3):120-5.
Mayer S, Mutschler E, Benet LZ, Sphahn-Langguth H. PMID: 8338721.
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PubMed Mentions: Fields:
Translation:
HumansCells
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Predictability of the covalent binding of acidic drugs in man. Life Sci. 1993; 53(8):PL141-6.
Benet LZ, Spahn-Langguth H, Iwakawa S, Volland C, Mizuma T, Mayer S, Mutschler E, Lin ET. PMID: 8350674.
View in:
PubMed Mentions:
15 Fields:
Translation:
HumansAnimalsCells
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Comparison of vasodilatory responses to nitroglycerin and its dinitrate metabolites in human veins. Clin Pharmacol Ther. 1992 Dec; 52(6):590-6.
Haefeli WE, Gumbleton M, Benet LZ, Hoffman BB, Blaschke TF. PMID: 1458768.
View in:
PubMed Mentions:
4 Fields:
Translation:
HumansCTClinical Trials
-
Glutathione S-transferase-mediated metabolism of glyceryl trinitrate in subcellular fractions of bovine coronary arteries. Pharm Res. 1992 Nov; 9(11):1460-4.
Lau DT, Chan EK, Benet LZ. PMID: 1475234.
View in:
PubMed Mentions:
6 Fields:
Translation:
AnimalsCells
-
Bioavailability of cyclosporine with concomitant rifampin administration is markedly less than predicted by hepatic enzyme induction. Clin Pharmacol Ther. 1992 Nov; 52(5):453-7.
Hebert MF, Roberts JP, Prueksaritanont T, Benet LZ. PMID: 1424418.
View in:
PubMed Mentions:
54 Fields:
Translation:
Humans
-
Elderly, conscious patients have an accentuated hypotensive response to nitroglycerin. Anesthesiology. 1992 Oct; 77(4):646-55.
Cahalan MK, Hashimoto Y, Aizawa K, Verotta D, Ionescu P, Balea M, Eger EI, Benet LZ, Ehrenfeld WK, Goldstone J, et al. PMID: 1416161.
View in:
PubMed Mentions:
5 Fields:
Translation:
HumansCTClinical Trials
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Improved gas chromatographic assay for the simultaneous determination of nitroglycerin and its mono- and dinitrate metabolites. J Chromatogr. 1992 Sep 02; 579(2):237-45.
Han C, Gumbleton M, Lau DT, Benet LZ. PMID: 1429971.
View in:
PubMed Mentions:
5 Fields:
Translation:
Humans
-
Effects of low-density lipoprotein and ethinyl estradiol on cyclosporine metabolism in isolated rat liver perfusions. Drug Metab Dispos. 1992 Jul-Aug; 20(4):547-52.
Prueksaritanont T, Hoener BA, Benet LZ. PMID: 1356733.
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PubMed Mentions:
4 Fields:
Translation:
Animals
-
Opportunities for integration of pharmacokinetics, pharmacodynamics, and toxicokinetics in rational drug development. Pharm Res. 1992 Jun; 9(6):826-33.
Peck CC, Barr WH, Benet LZ, Collins J, Desjardins RE, Furst DE, Harter JG, Levy G, Ludden T, Rodman JH, et al. PMID: 1409369.
View in:
PubMed Mentions:
7 Fields:
Translation:
HumansAnimals
-
Opportunities for integration of pharmacokinetics, pharmacodynamics, and toxicokinetics in rational drug development. J Pharm Sci. 1992 Jun; 81(6):605-10.
Peck CC, Barr WH, Benet LZ, Collins J, Desjardins RE, Furst DE, Harter JG, Levy G, Ludden T, Rodman JH, et al. PMID: 1355792.
View in:
PubMed Mentions:
10 Fields:
Translation:
HumansAnimals
-
Effects of sulfobromophthalein and ethacrynic acid on glyceryl trinitrate relaxation. Biochem Pharmacol. 1992 May 28; 43(10):2247-54.
Lau DT, Benet LZ. PMID: 1599510.
View in:
PubMed Mentions:
5 Fields:
Translation:
Animals
-
Transport and metabolism of cyclosporine in isolated rat hepatocytes. The effects of lipids. Biochem Pharmacol. 1992 May 08; 43(9):1997-2006.
Prueksaritanont T, Koike M, Hoener BA, Benet LZ. PMID: 1596287.
View in:
PubMed Mentions:
5 Fields:
Translation:
AnimalsCells
-
Opportunities for integration of pharmacokinetics, pharmacodynamics, and toxicokinetics in rational drug development. Clin Pharmacol Ther. 1992 Apr; 51(4):465-73.
Peck CC, Barr WH, Benet LZ, Collins J, Desjardins RE, Furst DE, Harter JG, Levy G, Ludden T, Rodman JH, et al. PMID: 1563216.
View in:
PubMed Mentions:
35 Fields:
Translation:
HumansAnimals
-
Cutaneous metabolism of nitroglycerin in vitro. II. Effects of skin condition and penetration enhancement. Pharm Res. 1992 Mar; 9(3):303-6.
Higo N, Hinz RS, Lau DT, Benet LZ, Guy RH. PMID: 1614960.
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PubMed Mentions:
4 Fields:
Translation:
Animals
-
Cutaneous metabolism of nitroglycerin in vitro. I. Homogenized versus intact skin. Pharm Res. 1992 Feb; 9(2):187-90.
Higo N, Hinz RS, Lau DT, Benet LZ, Guy RH. PMID: 1553339.
View in:
PubMed Mentions:
6 Fields:
Translation:
Animals
-
Acyl glucuronides revisited: is the glucuronidation process a toxification as well as a detoxification mechanism? Drug Metab Rev. 1992; 24(1):5-47.
Spahn-Langguth H, Benet LZ. PMID: 1555494.
View in:
PubMed Mentions:
44 Fields:
Translation:
HumansAnimalsCells
-
The interconversion of prednisone and prednisolone in human and rabbit organs in vitro is a function of tissue integrity. Pharmacology. 1992; 44(5):273-82.
Hale VG, Benet LZ. PMID: 1620723.
View in:
PubMed Mentions:
1 Fields:
Translation:
HumansAnimalsCells
-
Stereoselective degradation of the fenoprofen acyl glucuronide enantiomers and irreversible binding to plasma protein. Drug Metab Dispos. 1991 Nov-Dec; 19(6):1080-6.
Volland C, Sun H, Dammeyer J, Benet LZ. PMID: 1687014.
View in:
PubMed Mentions:
3 Fields:
Translation:
HumansAnimalsCells
-
Disposition of prednisone and prednisolone in the perfused rabbit liver: modeling hepatic metabolic processes. J Pharmacokinet Biopharm. 1991 Oct; 19(5):597-614.
Hale VG, Aizawa K, Sheiner LB, Benet LZ. PMID: 1783993.
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PubMed Mentions: Fields:
Translation:
Animals
-
Percutaneous penetration kinetics of nitroglycerin and its dinitrate metabolites across hairless mouse skin in vitro. Pharm Res. 1991 Oct; 8(10):1231-7.
Kikkoji T, Gumbleton M, Higo N, Guy RH, Benet LZ. PMID: 1796039.
View in:
PubMed Mentions:
3 Fields:
Translation:
Animals
-
Stereoselective disposition of carprofen, flunoxaprofen, and naproxen in rats. Drug Metab Dispos. 1991 Sep-Oct; 19(5):853-7.
Iwakawa S, Spahn H, Benet LZ, Lin ET. PMID: 1686227.
View in:
PubMed Mentions:
3 Fields:
Translation:
Animals
-
Prednisone and prednisolone interconversion in the rabbit utilizing unbound concentrations. Biopharm Drug Dispos. 1991 Aug-Sep; 12(6):467-77.
Hammarlund-Udenaes M, Benet LZ. PMID: 1932610.
View in:
PubMed Mentions:
1 Fields:
Translation:
AnimalsCells
-
Variable glyceryl dinitrate formation following infusions of glyceryl trinitrate at different vascular sites in the rat. Pharm Res. 1991 Jul; 8(7):877-82.
Nakashima E, Lau DT, Benet LZ. PMID: 1924138.
View in:
PubMed Mentions:
1 Fields:
Translation:
Animals
-
Nitroglycerin absorption from transdermal systems: formulation effects and metabolite concentrations. Pharm Res. 1991 Jun; 8(6):744-9.
Williams RL, Thakker KM, John V, Lin ET, Liang-Gee W, Benet LZ. PMID: 1905809.
View in:
PubMed Mentions:
8 Fields:
Translation:
Humans
-
Stereoselective disposition of ketoprofen in rats. Drug Metab Dispos. 1991 May-Jun; 19(3):717-8.
Iwakawa S, He XW, Hashimoto S, Volland C, Benet LZ, Lin ET. PMID: 1680643.
View in:
PubMed Mentions:
3 Fields:
Translation:
Animals
-
Rho Chi Lecture. Ideals and innovation: drugs, generics, the FDA, and the pharmacist. DICP. 1991 Apr; 25(4):427-30.
Benet LZ. PMID: 1926916.
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PubMed Mentions: Translation:
Humans
-
Drug metabolism and laboratory anesthetic protocols in the rat: examination of antipyrine pharmacokinetics. Pharm Res. 1991 Apr; 8(4):544-6.
Gumbleton M, Benet LZ. PMID: 1871056.
View in:
PubMed Mentions:
4 Fields:
Translation:
Animals
-
Pharmacokinetic studies of the nitroglycerin metabolites, 1,2- and 1,3- glyceryl dinitrates, in the rat. Biopharm Drug Dispos. 1991 Apr; 12(3):215-22.
Lau DT, Gumbleton M, Labisch C, Benet LZ. PMID: 1905575.
View in:
PubMed Mentions:
3 Fields:
Translation:
Animals
-
Pharmacological activity of the dinitrate metabolites of nitroglycerin following their oral administration to healthy volunteers. Br J Clin Pharmacol. 1991 Feb; 31(2):211-3.
Gumbleton M, Benet LZ. PMID: 1904752; PMCID: PMC1368399.
View in:
PubMed Mentions:
11 Fields:
Translation:
Humans
-
Prednisolone and prednisone exhibit linear extraction in the perfused rabbit liver. Drug Metab Dispos. 1991 Jan-Feb; 19(1):87-93.
Hale VG, Benet LZ. PMID: 1673428.
View in:
PubMed Mentions:
5 Fields:
Translation:
AnimalsCells
-
Safety and pharmacokinetics: colloidal bismuth subcitrate. Scand J Gastroenterol Suppl. 1991; 185:29-35.
Benet LZ. PMID: 1957122.
View in:
PubMed Mentions:
10 Fields:
Translation:
Humans
-
In vitro enantioselective glucuronidation of fenoprofen. Pharmacology. 1991; 43(2):53-60.
Volland C, Benet LZ. PMID: 1775510.
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PubMed Mentions: Fields:
Translation:
HumansAnimalsCells
-
Stereoselective analysis of fenoprofen and its metabolites. J Chromatogr. 1990 Dec 14; 534:127-38.
Volland C, Sun H, Benet LZ. PMID: 2094699.
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PubMed Mentions: Fields:
Translation:
Humans
-
Pharmacokinetics and pharmacodynamics of glyceryl trinitrate and its two dinitrate metabolites in conscious dogs. J Pharmacol Exp Ther. 1990 Dec; 255(3):1222-9.
Lee FW, Salmonson T, Metzler CH, Benet LZ. PMID: 2124621.
View in:
PubMed Mentions:
9 Fields:
Translation:
Animals
-
Report of the workshop on in vitro and in vivo testing and correlation for oral controlled/modified-release dosage forms. J Pharm Sci. 1990 Sep; 79(9):849-54.
Skelley JP, Amidon GL, Barr WH, Benet LZ, Carter JE, Robinson JR, Shah VP, Yacobi A. PMID: 1980308.
View in:
PubMed Mentions:
20 Fields:
-
Covalent binding of zomepirac glucuronide to proteins: evidence for a Schiff base mechanism. Drug Metab Dispos. 1990 Sep-Oct; 18(5):639-44.
Smith PC, Benet LZ, McDonagh AF. PMID: 1981713.
View in:
PubMed Mentions:
8 Fields:
Translation:
HumansAnimalsCells
-
Determination of soluble IL-2 receptors in kidney graft recipients--a 6-month follow-up. Transplant Proc. 1990 Aug; 22(4):1861-2.
Manfro RC, Pohanka E, Tomlanovich SJ, Benet LZ, Salvatierra O, Garovoy MR. PMID: 2389461.
View in:
PubMed Mentions: Fields:
Translation:
Humans
-
Effect of food on the pharmacokinetics of cyclosporine in healthy subjects following oral and intravenous administration. J Clin Pharmacol. 1990 Jul; 30(7):643-53.
Gupta SK, Manfro RC, Tomlanovich SJ, Gambertoglio JG, Garovoy MR, Benet LZ. PMID: 2391396.
View in:
PubMed Mentions:
23 Fields:
Translation:
Humans
-
Pharmacokinetics of nitroglycerin and its dinitrate metabolites over a thirtyfold range of oral doses. Clin Pharmacol Ther. 1990 May; 47(5):592-8.
Nakashima E, Rigod JF, Lin ET, Benet LZ. PMID: 2111749.
View in:
PubMed Mentions:
11 Fields:
Translation:
Humans
-
Nitroglycerin metabolism in subcellular fractions of rabbit liver. Dose dependency of glyceryl dinitrate formation and possible involvement of multiple isozymes of glutathione S-transferases. Drug Metab Dispos. 1990 May-Jun; 18(3):292-7.
Lau DT, Benet LZ. PMID: 1974188.
View in:
PubMed Mentions:
10 Fields:
Translation:
AnimalsCells
-
Absorption and disposition of a new low-dose combination formulation of hydrochlorothiazide and triamterene. Biopharm Drug Dispos. 1990 Apr; 11(3):233-43.
Williams RL, Lin ET, Liang-Gee W, Blume CD, Benet LZ. PMID: 2328310.
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PubMed Mentions: Fields:
Translation:
HumansCTClinical Trials
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Fetal uptake of intraamniotic digoxin in sheep. Pediatr Res. 1990 Mar; 27(3):282-5.
Hamamoto K, Iwamoto HS, Roman CM, Benet LZ, Rudolph AM. PMID: 2320396.
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PubMed Mentions: Fields:
Translation:
Animals
-
Stereoselective binding of the glucuronide conjugates of carprofen enantiomers to human serum albumin. Biochem Pharmacol. 1990 Mar 01; 39(5):949-53.
Iwakawa S, Spahn H, Benet LZ, Lin ET. PMID: 2310420.
View in:
PubMed Mentions:
7 Fields:
Translation:
HumansCells
-
The effect of acetaminophen on zidovudine metabolism in HIV-infected patients. J Acquir Immune Defic Syndr (1988). 1990; 3(7):691-4.
Steffe EM, King JH, Inciardi JF, Flynn NF, Goldstein E, Tonjes TS, Benet LZ. PMID: 2352121.
View in:
PubMed Mentions:
8 Fields:
Translation:
Humans
-
Irreversible binding of tolmetin glucuronic acid esters to albumin in vitro. Pharm Res. 1990 Jan; 7(1):21-7.
Munafo A, McDonagh AF, Smith PC, Benet LZ. PMID: 2300531.
View in:
PubMed Mentions:
3 Fields:
Translation:
HumansCells
-
High-fat meals increase the clearance of cyclosporine. Pharm Res. 1990 Jan; 7(1):46-8.
Gupta SK, Benet LZ. PMID: 2300535.
View in:
PubMed Mentions:
20 Fields:
Translation:
Humans
-
Comparative study of acetaminophen disposition in sheep at three developmental stages: the fetal, neonatal and adult periods. Dev Pharmacol Ther. 1990; 14(3):161-79.
Wang LH, Rudolph AM, Benet LZ. PMID: 2364855.
View in:
PubMed Mentions:
2 Fields:
Translation:
Animals
-
Effect of esterase inhibition on the disposition of zomepirac glucuronide and its covalent binding to plasma proteins in the guinea pig. J Pharmacol Exp Ther. 1990 Jan; 252(1):218-24.
Smith PC, McDonagh AF, Benet LZ. PMID: 2299592.
View in:
PubMed Mentions:
4 Fields:
Translation:
AnimalsCells
-
An integrated approach to pharmacokinetic analysis for linear mammillary systems in which input and exit may occur in/from any compartment. J Pharmacokinet Biopharm. 1989 Dec; 17(6):673-86.
Nakashima E, Benet LZ. PMID: 2635739.
View in:
PubMed Mentions:
4 Fields:
-
Pharmacokinetics of nicotinic acid-salicylic acid interaction. Clin Pharmacol Ther. 1989 Dec; 46(6):642-7.
Ding RW, Kolbe K, Merz B, de Vries J, Weber E, Benet LZ. PMID: 2598568.
View in:
PubMed Mentions:
10 Fields:
Translation:
Humans
-
Absorption kinetics of cyclosporine in healthy volunteers. Biopharm Drug Dispos. 1989 Nov-Dec; 10(6):591-6.
Gupta SK, Benet LZ. PMID: 2611359.
View in:
PubMed Mentions:
5 Fields:
Translation:
HumansCTClinical Trials
-
Determination of mean input time, mean residence time, and steady-state volume of distribution with multiple drug inputs. J Pharmacokinet Biopharm. 1989 Oct; 17(5):593-9.
Watari N, Benet LZ. PMID: 2614687.
View in:
PubMed Mentions:
9 Fields:
-
Simultaneous measurement of prednisone, prednisolone and 6 beta-hydroxyprednisolone in urine by high-performance liquid chromatography using dexamethasone as the internal standard. J Chromatogr. 1989 Sep 01; 493(2):421-3.
Teng RL, Benet LZ. PMID: 2584309.
View in:
PubMed Mentions: Fields:
-
Direct determination of diastereomeric carprofen glucuronides in human plasma and urine and preliminary measurements of stereoselective metabolic and renal elimination after oral administration of carprofen in man. Drug Metab Dispos. 1989 Jul-Aug; 17(4):414-9.
Iwakawa S, Suganuma T, Lee SF, Spahn H, Benet LZ, Lin ET. PMID: 2571482.
View in:
PubMed Mentions:
6 Fields:
Translation:
Humans
-
Application of clearance concepts to the assessment of exposure to lead in drinking water. Am J Public Health. 1989 Jul; 79(7):827-31.
Bois FY, Tozer TN, Zeise L, Benet LZ. PMID: 2735466; PMCID: PMC1349658.
View in:
PubMed Mentions:
3 Fields:
Translation:
HumansPHPublic Health
-
Lead exposure in children vs adults. Am J Public Health. 1989 Jul; 79(7):904.
Bois FY, Tozer TN, Benet LZ, Zeise L. PMID: 2735489; PMCID: PMC1349686.
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PubMed Mentions: Fields:
Translation:
HumansPHPublic Health
-
Prediction of the distribution volumes of cefazolin and tobramycin in obese children based on physiological pharmacokinetic concepts. Pharm Res. 1989 Jun; 6(6):486-91.
Koshida R, Nakashima E, Taniguchi N, Tsuji A, Benet LZ, Ichimura F. PMID: 2762224.
View in:
PubMed Mentions:
14 Fields:
Translation:
HumansCells
-
Probenecid-induced changes in the clearance of carprofen enantiomers: a preliminary study. Clin Pharmacol Ther. 1989 May; 45(5):500-5.
Spahn H, Spahn I, Benet LZ. PMID: 2721105.
View in:
PubMed Mentions:
15 Fields:
Translation:
Humans
-
Differential effects of the degree of renal damage on p-aminohippuric acid and inulin clearances in rats. J Pharmacokinet Biopharm. 1989 Apr; 17(2):169-77.
Gloff CA, Benet LZ. PMID: 2795454.
View in:
PubMed Mentions:
11 Fields:
Translation:
Animals
-
Furosemide pharmacokinetics and pharmacodynamics in health and disease--an update. J Pharmacokinet Biopharm. 1989 Feb; 17(1):1-46.
Hammarlund-Udenaes M, Benet LZ. PMID: 2654356.
View in:
PubMed Mentions:
29 Fields:
Translation:
Humans
-
Procedures to characterize in vivo and in vitro enantioselective glucuronidation properly: studies with benoxaprofen glucuronides. Pharm Res. 1989 Feb; 6(2):125-32.
Spahn H, Iwakawa S, Lin ET, Benet LZ. PMID: 2762212.
View in:
PubMed Mentions:
4 Fields:
Translation:
HumansAnimalsCells
-
Differential formation of dinitrate metabolites from glyceryl trinitrate in subcellular fractions of rabbit liver. Biochem Pharmacol. 1989 Feb 01; 38(3):543-6.
Lau DT, Benet LZ. PMID: 2492808.
View in:
PubMed Mentions:
4 Fields:
Translation:
AnimalsCells
-
Cyclosporin A and prednisolone: an additive inhibitory effect of cell proliferation and interleukin-2 production. Transplant Proc. 1989 Feb; 21(1 Pt 2):1457-9.
Manfro RC, Pohanka E, Tomlanovich S, Benet LZ, Garovoy MR. PMID: 2523586.
View in:
PubMed Mentions:
2 Fields:
Translation:
HumansCells
-
Measurement of carprofen enantiomer concentrations in plasma and urine using L-leucinamide as the chiral coupling component. J Chromatogr. 1988 Dec 09; 433:331-8.
Spahn H, Spahn I, Pflugmann G, Mutschler E, Benet LZ. PMID: 3235564.
View in:
PubMed Mentions:
1 Fields:
Translation:
Humans
-
Pharmacokinetics of nitroglycerin and metabolites in humans following oral dosing. Biopharm Drug Dispos. 1988 Nov-Dec; 9(6):557-65.
Yu DK, Williams RL, Benet LZ, Lin ET, Giesing DH. PMID: 3147725.
View in:
PubMed Mentions:
13 Fields:
Translation:
Humans
-
General treatment of mean residence time, clearance, and volume parameters in linear mammillary models with elimination from any compartment. J Pharmacokinet Biopharm. 1988 Oct; 16(5):475-92.
Nakashima E, Benet LZ. PMID: 3199315.
View in:
PubMed Mentions:
16 Fields:
Translation:
Humans
-
Ion-paired liquid chromatographic method for the analysis of blood and plasma for the antimalarial drug halofantrine and its putative mono-debutylated metabolite. J Chromatogr. 1988 Sep 09; 430(2):412-9.
Gawienowski M, Benet LZ, Fleckenstein L, Lin ET. PMID: 3235515.
View in:
PubMed Mentions:
2 Fields:
Translation:
Humans
-
Disposition and irreversible plasma protein binding of tolmetin in humans. Clin Pharmacol Ther. 1988 Jul; 44(1):107-14.
Hyneck ML, Smith PC, Munafo A, McDonagh AF, Benet LZ. PMID: 3390998.
View in:
PubMed Mentions:
11 Fields:
Translation:
Humans
-
Effect of cimetidine or ranitidine administration on nifedipine pharmacokinetics and pharmacodynamics. Clin Pharmacol Ther. 1988 Jun; 43(6):673-80.
Schwartz JB, Upton RA, Lin ET, Williams RL, Benet LZ. PMID: 3378388.
View in:
PubMed Mentions:
15 Fields:
Translation:
Humans
-
Simultaneous determination of nitroglycerin and its dinitrate metabolites by capillary gas chromatography with electron-capture detection. J Chromatogr. 1988 Apr 29; 426(2):259-66.
Lee FW, Watari N, Rigod J, Benet LZ. PMID: 3134385.
View in:
PubMed Mentions:
9 Fields:
Translation:
HumansAnimals
-
Effect of pH on acyl migration and hydrolysis of tolmetin glucuronide. Drug Metab Dispos. 1988 Mar-Apr; 16(2):322-4.
Hyneck ML, Munafo A, Benet LZ. PMID: 2898354.
View in:
PubMed Mentions:
4 Fields:
Translation:
HumansCells
-
Organic anion transport by basal-lateral membranes: effect of PAH and furosemide on each other's transport. Pharmacology. 1988; 37(4):268-76.
Gloff CA, Mamelok RD, Benet LZ. PMID: 3194444.
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PubMed Mentions: Fields:
Translation:
AnimalsCells
-
High-performance liquid chromatographic determination of tolmetin, tolmetin glucuronide and its isomeric conjugates in plasma and urine. J Chromatogr. 1987 Sep 25; 420(2):349-56.
Hyneck ML, Smith PC, Unseld E, Benet LZ. PMID: 3693506.
View in:
PubMed Mentions:
4 Fields:
Translation:
HumansCells
-
Variable glyceryl dinitrate formation as a function of route of nitroglycerin administration. Clin Pharmacol Ther. 1987 Sep; 42(3):273-7.
Noonan PK, Benet LZ. PMID: 3113806.
View in:
PubMed Mentions:
12 Fields:
Translation:
Humans
-
Transdermal bioavailability and first-pass skin metabolism: a preliminary evaluation with nitroglycerin. J Pharmacokinet Biopharm. 1987 Aug; 15(4):423-37.
Nakashima E, Noonan PK, Benet LZ. PMID: 3119815.
View in:
PubMed Mentions:
10 Fields:
Translation:
Humans
-
Effects of formulation and food on the absorption of hydrochlorothiazide and triamterene or amiloride from combination diuretic products. Pharm Res. 1987 Aug; 4(4):348-52.
Williams RL, Mordenti J, Upton RA, Lin ET, Gee WL, Blume CD, Benet LZ. PMID: 3508542.
View in:
PubMed Mentions:
5 Fields:
Translation:
Humans
-
Pharmacokinetics and excretion of unique beta-adrenergic agonists. Pharmacology. 1987; 34(2-3):157-66.
Ferraiolo BL, Halldin MM, Asscher Y, Akita Y, Melmon KL, Benet LZ, Castagnoli N. PMID: 2884679.
View in:
PubMed Mentions: Fields:
Translation:
Animals
-
Developmental alterations in hepatic UDP-glucuronosyltransferase. A comparison of the kinetic properties of enzymes from adult sheep and fetal lambs. Biochem Pharmacol. 1986 Sep 15; 35(18):3065-70.
Wang LH, Zakim D, Rudolph AM, Benet LZ. PMID: 3092831.
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PubMed Mentions: Fields:
Translation:
Animals
-
Absorption and disposition of two combination formulations of hydrochlorothiazide and triamterene: influence of age and renal function. Clin Pharmacol Ther. 1986 Aug; 40(2):226-32.
Williams RL, Thornhill MD, Upton RA, Blume C, Clark TS, Lin E, Benet LZ. PMID: 3731685.
View in:
PubMed Mentions:
4 Fields:
Translation:
HumansCells
-
AAPS and pharmaceutical research. Pharm Res. 1986 Aug; 3(4):186.
Benet LZ. PMID: 24271580.
View in:
PubMed Mentions: Fields:
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Pharmacokinetic studies of the disposition of acetaminophen in the sheep maternal-placental-fetal unit. J Pharmacol Exp Ther. 1986 Jul; 238(1):198-205.
Wang LH, Rudolph AM, Benet LZ. PMID: 3723398.
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PubMed Mentions:
7 Fields:
Translation:
Animals
-
Ethambutol kinetics in patients with impaired renal function. Am Rev Respir Dis. 1986 Jul; 134(1):34-8.
Varughese A, Brater DC, Benet LZ, Lee CS. PMID: 3729159.
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PubMed Mentions:
12 Fields:
Translation:
Humans
-
Characterization of the isomeric esters of zomepirac glucuronide by proton NMR. Drug Metab Dispos. 1986 Jul-Aug; 14(4):503-5.
Smith PC, Benet LZ. PMID: 2874000.
View in:
PubMed Mentions:
3 Fields:
Translation:
HumansCells
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High-performance liquid chromatographic assay of basic amine drugs in plasma and urine using a silica gel column and an aqueous mobile phase. I. Amiloride. J Chromatogr. 1986 Apr 25; 377:399-404.
Shi RJ, Benet LZ, Lin ET. PMID: 3711234.
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PubMed Mentions: Fields:
Translation:
Humans
-
Marked alterations in dose-dependent prednisolone kinetics in women taking oral contraceptives. Clin Pharmacol Ther. 1986 Apr; 39(4):425-9.
Legler UF, Benet LZ. PMID: 3956058.
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PubMed Mentions:
7 Fields:
Translation:
Humans
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Irreversible binding of zomepirac to plasma protein in vitro and in vivo. J Clin Invest. 1986 Mar; 77(3):934-9.
Smith PC, McDonagh AF, Benet LZ. PMID: 3949982; PMCID: PMC423485.
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PubMed Mentions:
15 Fields:
Translation:
HumansCells
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The bioavailability of oral nitroglycerin. J Pharm Sci. 1986 Mar; 75(3):241-3.
Noonan PK, Benet LZ. PMID: 3084757.
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PubMed Mentions:
14 Fields:
Translation:
Humans
-
Metabolic fate and solubility of triamterene--not an explanation for triamterene nephrolithiasis. J Pharm Sci. 1986 Feb; 75(2):129-32.
Sörgel F, Ettinger B, Benet LZ. PMID: 3958920.
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PubMed Mentions:
1 Fields:
Translation:
Humans
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The effect of prednisone and hydrocortisone on the plasma protein binding of prednisolone in man. Eur J Clin Pharmacol. 1986; 30(1):51-5.
Legler UF, Benet LZ. PMID: 3709632.
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PubMed Mentions:
5 Fields:
Translation:
HumansCells
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Impairment of prednisolone disposition in women taking oral contraceptives or conjugated estrogens. J Clin Endocrinol Metab. 1986 Jan; 62(1):234-7.
Gustavson LE, Legler UF, Benet LZ. PMID: 2999180.
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PubMed Mentions:
9 Fields:
Translation:
Humans
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The macromolecular binding of prednisone in plasma of healthy volunteers including pregnant women and oral contraceptive users. J Pharmacokinet Biopharm. 1985 Dec; 13(6):561-9.
Gustavson LE, Benet LZ. PMID: 3834071.
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PubMed Mentions:
3 Fields:
Translation:
HumansCells
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Premarketing observational studies of population pharmacokinetics of new drugs. Clin Pharmacol Ther. 1985 Nov; 38(5):481-7.
Sheiner LB, Benet LZ. PMID: 3931953.
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PubMed Mentions:
28 Fields:
Translation:
HumansCTClinical Trials
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Distribution and fate of acetaminophen conjugates in fetal lambs in utero. J Pharmacol Exp Ther. 1985 Nov; 235(2):302-7.
Wang LH, Rudolph AM, Benet LZ. PMID: 4057072.
View in:
PubMed Mentions:
2 Fields:
Translation:
Animals
-
Mean residence time in the body versus mean residence time in the central compartment. J Pharmacokinet Biopharm. 1985 Oct; 13(5):555-8.
Benet LZ. PMID: 3834069.
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PubMed Mentions:
10 Fields:
Translation:
HumansPHPublic Health
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Effect of probenecid on the formation and elimination of acyl glucuronides: studies with zomepirac. Clin Pharmacol Ther. 1985 Aug; 38(2):121-7.
Smith PC, Langendijk PN, Bosso JA, Benet LZ. PMID: 3874742.
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PubMed Mentions:
17 Fields:
Translation:
Humans
-
Peptides and proteins as drugs. Pharm Res. 1985 Jul; 2(4):151-6.
Ferraiolo BL, Benet LZ. PMID: 24272804.
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PubMed Mentions:
3 Fields:
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Dose dependent pharmacokinetics of nitroglycerin after multiple intravenous infusions in healthy volunteers. J Pharmacokinet Biopharm. 1985 Apr; 13(2):143-57.
Noonan PK, Williams RL, Benet LZ. PMID: 3932639.
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PubMed Mentions:
18 Fields:
Translation:
HumansCells
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Pharmacokinetics and metabolism of bepridil. Am J Cardiol. 1985 Mar 15; 55(7):8C-13C.
Benet LZ. PMID: 3872057.
View in:
PubMed Mentions:
8 Fields:
Translation:
HumansAnimalsCells
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Pharmacokinetics of drugs and metabolites in the maternal-placental-fetal unit: general principles. NIDA Res Monogr. 1985; 60:25-38.
Wang LH, Rudolph AM, Benet LZ. PMID: 3932864.
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PubMed Mentions:
1 Fields:
Translation:
Humans
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Incomplete and delayed bioavailability of sublingual nitroglycerin. Am J Cardiol. 1985 Jan 01; 55(1):184-7.
Noonan PK, Benet LZ. PMID: 3917598.
View in:
PubMed Mentions:
16 Fields:
Translation:
Humans
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Stability of acyl glucuronides in blood, plasma, and urine: studies with zomepirac. Drug Metab Dispos. 1985 Jan-Feb; 13(1):110-2.
Smith PC, Hasegawa J, Langendijk PN, Benet LZ. PMID: 2858367.
View in:
PubMed Mentions:
11 Fields:
Translation:
HumansAnimals
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Immunosuppressive activity of prednisone and prednisolone and their metabolic interconversion in the mixed lymphocyte reaction. Int J Immunopharmacol. 1985; 7(5):731-7.
Tsang SY, Garovoy MR, Benet LZ. PMID: 2931388.
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PubMed Mentions:
2 Fields:
Translation:
Humans
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Absence of a significant pharmacokinetic interaction between hydrochlorothiazide and triamterene when coadministered. J Pharmacokinet Biopharm. 1984 Dec; 12(6):575-86.
Upton RA, Williams RL, Lin ET, Gee WL, Blume CD, Benet LZ. PMID: 6533293.
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PubMed Mentions:
2 Fields:
Translation:
HumansCells
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Bioequivalence study of a new tablet formulation of triamterene and hydrochlorothiazide. Am J Med. 1984 Nov 05; 77(5A):59-61.
Blume CD, Williams RL, Upton RA, Lin ET, Benet LZ. PMID: 6496560.
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PubMed Mentions:
4 Fields:
Translation:
HumansCTClinical Trials
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Determination of picogram nitroglycerin plasma concentrations using capillary gas chromatography with on-column injection. J Pharm Sci. 1984 Jul; 73(7):923-7.
Noonan PK, Kanfer I, Riegelman S, Benet LZ. PMID: 6432997.
View in:
PubMed Mentions:
4 Fields:
Translation:
Humans
-
Liquid chromatographic analysis of triamterene and its major metabolite, hydroxytriamterene sulfate, in blood, plasma, and urine. J Pharm Sci. 1984 Jun; 73(6):831-3.
Sörgel F, Lin ET, Hasegawa J, Benet LZ. PMID: 6737274.
View in:
PubMed Mentions:
2 Fields:
Translation:
Humans
-
Simultaneous determination of zomepirac and its major metabolite zomepirac glucuronide in human plasma and urine. J Chromatogr. 1984 May 11; 307(2):371-9.
Langendijk PN, Smith PC, Hasegawa J, Benet LZ. PMID: 6610684.
View in:
PubMed Mentions:
3 Fields:
Translation:
Humans
-
High-performance liquid chromatographic method for the determination of indomethacin and its two primary metabolites in urine. J Chromatogr. 1984 Mar 09; 306:315-21.
Smith PC, Benet LZ. PMID: 6715469.
View in:
PubMed Mentions:
3 Fields:
Translation:
Humans
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Pharmacokinetic parameters: which are necessary to define a drug substance? Eur J Respir Dis Suppl. 1984; 134:45-61.
Benet LZ. PMID: 6586486.
View in:
PubMed Mentions:
7 Fields:
Translation:
Humans
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Unchanged absorption of digoxin tablets in patients with cardiac failure. Pharmacology. 1984; 28(2):90-4.
Meister W, Benowitz NL, Benet LZ. PMID: 6709691.
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PubMed Mentions: Fields:
Translation:
HumansCells
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Dose-dependent kinetics of probenecid in rhesus monkeys--infusion studies. Pharmacology. 1984; 28(4):181-7.
Chiang CW, Benet LZ. PMID: 6728896.
View in:
PubMed Mentions:
4 Fields:
Translation:
Animals
-
Oral bioavailability and intravenous pharmacokinetics of amrinone in humans. J Pharm Sci. 1983 Jul; 72(7):817-9.
Park GB, Kershner RP, Angellotti J, Williams RL, Benet LZ, Edelson J. PMID: 6886991.
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PubMed Mentions:
10 Fields:
Translation:
Humans
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Dose-dependent bioavailability of prazosin in beagle dogs. J Cardiovasc Pharmacol. 1983 Jul-Aug; 5(4):613-7.
Baughman RA, Sorgel F, Mico BA, Benet LZ. PMID: 6193359.
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PubMed Mentions: Fields:
Translation:
Animals
-
Prednisolone clearance: a possible determinant for glucocorticoid efficacy in patients with oral vesiculo-erosive diseases. J Dent Res. 1983 May; 62(5):575-7.
Lozada F, Frey FJ, Benet LZ. PMID: 6573375.
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PubMed Mentions:
1 Fields:
Translation:
Humans
-
Furosemide assays and disposition in healthy volunteers and renal transplant patients. Fed Proc. 1983 Apr; 42(6):1695-8.
Benet LZ, Smith DE, Lin ET, Vincenti F, Gambertoglio JG. PMID: 6339277.
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PubMed Mentions:
4 Fields:
Translation:
Humans
-
The bioavailability and disposition of tiodazosin levulinate in beagle dogs with a comparison to prazosin hydrochloride. Drug Metab Dispos. 1983 Mar-Apr; 11(2):143-6.
Baughman RA, Mico BA, Benet LZ. PMID: 6133719.
View in:
PubMed Mentions:
1 Fields:
Translation:
Animals
-
Biotransformation of furosemide in kidney transplant patients. Eur J Clin Pharmacol. 1983; 24(6):787-90.
Smith DE, Benet LZ. PMID: 6350024.
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PubMed Mentions:
10 Fields:
Translation:
Humans
-
Plasma protein binding of furosemide in kidney transplant patients. J Pharmacokinet Biopharm. 1982 Dec; 10(6):663-74.
Smith DE, Benet LZ. PMID: 6763626.
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PubMed Mentions:
5 Fields:
Translation:
HumansCells
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Endogenous and exogenous glucocorticoids in cushingoid patients. Drug Intell Clin Pharm. 1982 Nov; 16(11):863-8.
Benet LZ, Frey FJ, Amend WJ, Lozada F, Frey BM. PMID: 6756849.
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PubMed Mentions:
5 Fields:
Translation:
HumansCells
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Prednisolone clearance at steady state in man. J Clin Endocrinol Metab. 1982 Oct; 55(4):762-7.
Legler UF, Frey FJ, Benet LZ. PMID: 7107818.
View in:
PubMed Mentions:
16 Fields:
Translation:
Humans
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Pharmacokinetics of triamterene and its metabolite in man. J Pharmacokinet Biopharm. 1982 Oct; 10(5):507-23.
Hasegawa J, Lin ET, Williams RL, Sörgel F, Benet LZ. PMID: 7166735.
View in:
PubMed Mentions:
7 Fields:
Translation:
HumansCells
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Disposition of zomepirac sodium in man. J Clin Pharmacol. 1982 Oct; 22(10):470-6.
O'Neill PJ, Yorgey KA, Renzi NL, Williams RL, Benet LZ. PMID: 7174855.
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PubMed Mentions:
1 Fields:
Translation:
HumansCells
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Apparent intramolecular acyl migration of zomepirac glucuronide. Drug Metab Dispos. 1982 Sep-Oct; 10(5):469-73.
Hasegawa J, Smith PC, Benet LZ. PMID: 6128195.
View in:
PubMed Mentions:
11 Fields:
Translation:
Humans
-
Specific and sensitive assay of celiprolol in blood, plasma and urine using high-performance liquid chromatography. J Chromatogr. 1982 Jul 09; 230(2):454-60.
Buskin JN, Upton RA, Sörgel F, Williams RL, Lang E, Benet LZ. PMID: 6213630.
View in:
PubMed Mentions:
3 Fields:
Translation:
Humans
-
Determination of tiodazosin in plasma and whole blood by high-performance liquid chromatography. J Chromatogr. 1982 Jun 11; 230(1):203-6.
Mico BA, Baughman RA, Benet LZ. PMID: 7107763.
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PubMed Mentions: Fields:
Translation:
Animals
-
Prednisolone pharmacodynamics assessed by inhibition of the mixed lymphocyte reaction. Transplantation. 1982 Jun; 33(6):578-84.
Frey BM, Frey FJ, Holford NH, Lozada F, Benet LZ. PMID: 6213074.
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PubMed Mentions:
12 Fields:
Translation:
HumansCells
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Relative bioavailability of chlorthalidone in humans: adverse influence of polyethylene glycol. J Pharm Sci. 1982 May; 71(5):533-5.
Williams RL, Blume CD, Lin ET, Holford NH, Benet LZ. PMID: 7097499.
View in:
PubMed Mentions:
2 Fields:
Translation:
Humans
-
Hydrochlorothiazide pharmacokinetics and pharmacologic effect: the influence of indomethacin. J Clin Pharmacol. 1982 Jan; 22(1):32-41.
Williams RL, Davies RO, Berman RS, Holmes GI, Huber P, Gee WL, Lin ET, Benet LZ. PMID: 7061724.
View in:
PubMed Mentions:
3 Fields:
Translation:
Humans
-
Nonlinear plasma protein binding and haemodialysis clearance of prednisolone. Eur J Clin Pharmacol. 1982; 23(1):65-74.
Frey FJ, Gambertoglio JG, Frey BM, Benet LZ, Amend WJ. PMID: 6751835.
View in:
PubMed Mentions:
8 Fields:
Translation:
HumansCells
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Endogenous hydrocortisone, a possible factor contributing to the genesis of cushingoid habitus in patients on prednisone. J Clin Endocrinol Metab. 1981 Nov; 53(5):1076-80.
Frey FJ, Amend WJ, Lozada F, Frey BM, Benet LZ. PMID: 7026594.
View in:
PubMed Mentions:
7 Fields:
Translation:
Humans
-
Effects of indomethacin and carprofen on renal homeostasis in rheumatoid arthritis patients and in healthy individuals. J Clin Pharmacol. 1981 Nov-Dec; 21(11):493-500.
Williams RL, Furst DE, Mandel HG, Nicoll D, Konikoff JJ, Benet LZ. PMID: 7037867.
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PubMed Mentions: Fields:
Translation:
Humans
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Membrane populations of bovine choroid plexus: separation by density gradient centrifugation in modified colloidal silica. J Neurochem. 1981 Sep; 37(3):768-74.
Mamelok RD, Macrae DR, Benet LZ, Prusiner SB. PMID: 6115891.
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PubMed Mentions: Fields:
Translation:
AnimalsCells
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Saturable kinetics of intravenous chlorothiazide in the rhesus monkey. J Pharmacokinet Biopharm. 1981 Aug; 9(4):461-76.
Gustafson JH, Benet LZ. PMID: 7310644.
View in:
PubMed Mentions:
3 Fields:
Translation:
AnimalsCells
-
Furosemide kinetics and dynamics after kidney transplant. Clin Pharmacol Ther. 1981 Jul; 30(1):105-13.
Smith DE, Gambertoglio JG, Vincenti F, Benet LZ. PMID: 7016396.
View in:
PubMed Mentions:
12 Fields:
Translation:
Humans
-
A standard approach to compiling clinical pharmacokinetic data. J Pharmacokinet Biopharm. 1981 Feb; 9(1):59-127.
Sheiner LB, Benet LZ, Pagliaro LA. PMID: 7014827.
View in:
PubMed Mentions:
11 Fields:
Translation:
Humans
-
Dose-dependent kinetics of probenecid in rhesus monkeys-intravenous bolus studies. Pharmacology. 1981; 23(6):326-36.
Chiang CW, Benet LZ. PMID: 7312942.
View in:
PubMed Mentions:
2 Fields:
Translation:
AnimalsCells
-
Pharmacokinetics of prednisolone and endogenous hydrocortisone levels in cushingoid and non-cushingoid patients. Eur J Clin Pharmacol. 1981; 21(3):235-42.
Frey FJ, Amend WJ, Lozada F, Frey BM, Holford NH, Benet LZ. PMID: 7032949.
View in:
PubMed Mentions:
16 Fields:
Translation:
HumansCTClinical Trials
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Induction kinetics of human suppressor cells in the mixed lymphocyte reaction and influence of prednisolone on their genesis. Cell Immunol. 1980 Nov; 56(1):225-34.
Frey BM, Frey FJ, Cochrum KC, Benet LZ. PMID: 6448699.
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PubMed Mentions: Fields:
Translation:
HumansCells
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Renal excretion of pseudoephedrine. Clin Pharmacol Ther. 1980 Nov; 28(5):690-4.
Brater DC, Kaojarern S, Benet LZ, Lin ET, Lockwood T, Morris RC, McSherry EJ, Melmon KL. PMID: 7438686.
View in:
PubMed Mentions:
4 Fields:
Translation:
Humans
-
Prednisolone clearance at steady state in dogs. J Pharmacol Exp Ther. 1980 Nov; 215(2):287-91.
Frey FJ, Frey BM, Greither A, Benet LZ. PMID: 7441495.
View in:
PubMed Mentions:
21 Fields:
Translation:
HumansAnimals
-
High-performance liquid chromatographic determination of prazosin in human plasma, whole blood and urine. J Chromatogr. 1980 Sep 12; 183(3):367-71.
Lin ET, Baughman RA, Benet LZ. PMID: 7419656.
View in:
PubMed Mentions:
4 Fields:
Translation:
Humans
-
Absorption and disposition of furosemide in healthy volunteers, measured with a metabolite-specific assay. Drug Metab Dispos. 1980 Sep-Oct; 8(5):337-42.
Smith DE, Lin ET, Benet LZ. PMID: 6107232.
View in:
PubMed Mentions:
29 Fields:
Translation:
HumansCellsCTClinical Trials
-
Disposition kinetics of ethambutol in man. J Pharmacokinet Biopharm. 1980 Aug; 8(4):335-46.
Lee CS, Brater DC, Gambertoglio JG, Benet LZ. PMID: 7431225.
View in:
PubMed Mentions:
20 Fields:
Translation:
HumansCells
-
Altered prazosin pharmacokinetics in congestive heart failure. Eur J Clin Pharmacol. 1980 Jun; 17(6):425-8.
Baughman RA, Arnold S, Benet LZ, Lin ET, Chatterjee K, Williams RL. PMID: 7398734.
View in:
PubMed Mentions:
9 Fields:
Translation:
Humans
-
Preliminary evaluation of furosemide-probenecid interaction in humans. J Pharm Sci. 1980 May; 69(5):571-5.
Smith DE, Gee WL, Brater DC, Lin ET, Benet LZ. PMID: 7381747.
View in:
PubMed Mentions:
17